| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HSD11B2 |
(1S,4S,7R,9S)-7,8,9-trihydroxy-8-methyl-1-propan-2-ylspiro[4.5]decane-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1S,4S,5S)-8-methyl-9-oxo-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1R,4R,5R,9R)-9-hydroxy-8-methyl-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1R,4S,5S,9S)-9-hydroxy-1-methyl-8-methylidenespiro[4.5]decane-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1S,4S,5S,10R)-10-hydroxy-8-methyl-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1S,4S,5S,8S,9S)-1-cyclohexyl-8,9-dihydroxy-8-methylspiro[4.5]decane-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1S,4S,5S,9S)-9-hydroxy-8-methyl-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
(1S,4S,5S,9S)-9-acetyloxy-8-methyl-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
2-(Phenylsulfonyl)-1-p-tolylethanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
1-(3-Methoxyphenyl)-2-(phenylsulfonyl)ethanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
N-(6-aminopyridin-2-yl)-4'-cyanobiphenyl-4-sulfonamide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
Colletoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
methyl (1S,4S,5S,9S)-9-hydroxy-8-methyl-1-propan-2-ylspiro[4.5]dec-7-ene-4-carboxylate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
4'-Methoxy-2-(phenylsulfonyl)acetophenone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
4-[(3-Chlorophenylsulfonamido)methyl]-N-cycloheptyl-N-propylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
N-(4-phenyloxazol-2-yl)benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
3-Chloro-2-methyl-N-(4-phenyl-oxazol-2-yl)-benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
3-chloro-N-(4-(4-cyanophenyl)oxazol-2-yl)-2-methylbenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
N-[4-(4,5-Dimethyl-oxazol-2-ylsulfamoyl)-phenyl]-N-methyl-acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HSD11B2 |
4-[(3-Chlorophenylsulfonamido)methyl]-N-(1-adamantyl)benzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |