GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
AADAT |
HGNC:17929 |
Q8N5Z0 |
(3S)-3-amino-6-benzyl-1-hydroxy-7-methoxy-3,4-dihydroquinolin-2-one |
59627033 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
(3S)-3-amino-1-hydroxy-5-(trifluoromethyl)-3,4-dihydroquinolin-2-one |
62707349 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
(5S)-5-amino-7-hydroxy-2-phenyl-4,5-dihydropyrazolo[3,4-b]pyridin-6-one |
67813781 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
(3S)-3-amino-1-hydroxy-7-methoxy-6-phenoxy-3,4-dihydroquinolin-2-one |
71717990 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
US10065972, Example 579 |
124153855 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
US10065972, Example 565 |
124154150 |
BindingDB |
AADAT |
HGNC:17929 |
Q8N5Z0 |
2-cyclopropyl-N-(4-methoxyphenyl)-3-oxo-2,8-diazaspiro[5.5]undecane-8-carboxamide |
156010411 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Imatinib |
5291 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Staurosporine |
44259 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Gefitinib |
123631 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Vatalanib |
151194 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Canertinib |
156414 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Doramapimod |
156422 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Seliciclib |
160355 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole |
176155 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Lapatinib |
208908 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Sorafenib |
216239 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
6-(2,6-dichlorophenyl)-8-methyl-2-((3-(methylthio)phenyl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one |
447077 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
451705 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Nilotinib |
644241 |
BindingDB |