GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
AAK1 |
HGNC:19679 |
Q2M2I8 |
2-Cycloheptyl-4-[4-methoxy-3-(5-phenylpentoxy)phenyl]-4a,5,8,8a-tetrahydrophthalazin-1-one |
11113983 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Brivanib |
11234052 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
4-(2,6-dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide |
11338033 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Ast-487 |
11409972 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Linifanib |
11485656 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
GW-2580 |
11617559 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Raf-265 |
11656518 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Motesanib |
11667893 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
4-[[9-Chloro-7-(2,6-difluorophenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]benzoic acid |
11712649 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
(R)-5-(6-((4-methylpiperazin-1-yl)methyl)-1H-benzo[d]imidazol-1-yl)-3-(1-(2-(trifluoromethyl)phenyl)ethoxy)thiophene-2-carboxamide |
15983966 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Azd-1152hqpa |
16007391 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Gsk-690693 |
16725726 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
N-(3-(5-chloro-1H-pyrrolo[2,3-b]pyridine-3-carbonyl)-2,4-difluorophenyl)propane-1-sulfonamide |
24180719 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Quizartinib |
24889392 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
Ruxolitinib |
25126798 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
2-((2-((1-(2-(Dimethylamino)acetyl)-5-methoxyindolin-6-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-6-fluoro-N-methylbenzamide |
25182616 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
1-N-(4-fluorocyclohexa-1,5-dien-1-yl)-1-N'-[3-fluoro-4-[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxyphenyl]cyclopropane-1,1-dicarboxamide |
57399640 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
(S)-8-((2-amino-4-methylpentyl)oxy)-4,6-dimethyl-5-oxo-5,6-dihydrobenzo[c][2,7]naphthyridine-9-carbonitrile |
73214233 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
N-(5H-chromeno[3,4-c]pyridin-8-yl)-3-isopropylpiperidine-2-carboxamide |
78324812 |
BindingDB |
AAK1 |
HGNC:19679 |
Q2M2I8 |
2-{4-[(1Z)-1-(hydroxyimino)-2,3-dihydro-1H-inden-5-yl]-3-(pyridin-4-yl)-1H-pyrazol-1-yl}ethan-1-ol |
91448975 |
BindingDB |