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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA2A HGNC:263 P29274 1,3-dipropyl-8-(1-((3-(4-(trifluoromethyl)phenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1H-purine-2,6(3H,7H)-dione 44406639 BindingDB
ADORA2A HGNC:263 P29274 4-(5-((4-(2,6-dioxo-1,3-dipropyl-2,3,6,7-tetrahydro-1H-purin-8-yl)-1H-pyrazol-1-yl)methyl)-1,2,4-oxadiazol-3-yl)benzonitrile 44406642 BindingDB
ADORA2A HGNC:263 P29274 8-(1-((3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione 44406643 BindingDB
ADORA2A HGNC:263 P29274 8-[6-[2-(4-iodophenyl)-2-oxoethoxy]pyridazin-3-yl]-1,3-dipropyl-7H-purine-2,6-dione 44406904 BindingDB
ADORA2A HGNC:263 P29274 8-[5-[2-(4-iodophenyl)-2-oxoethoxy]pyridin-2-yl]-1,3-dipropyl-7H-purine-2,6-dione 44406920 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-[2-(dimethylamino)-6-[(3-iodophenyl)methylamino]purin-9-yl]-3,4-dihydroxy-N,N-dimethyloxolane-2-carboxamide 44407518 BindingDB
ADORA2A HGNC:263 P29274 (2R,3R,4S,5R)-2-(6-amino-2-(2-(thiophen-2-yl)ethoxy)-9H-purin-9-yl)-5-(hydroxymethyl)-tetrahydrofuran-3,4-diol 44420921 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-oxo-2-(phenylamino)ethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 44423811 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-5-(6-(4-(2-(4-fluorophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423812 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(4-chlorophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423813 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(4-bromophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423814 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-iodophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 44423815 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-[6-[4-[2-oxo-2-[2-(trifluoromethyl)anilino]ethoxy]anilino]purin-9-yl]oxolane-2-carboxamide 44423816 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-methoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 44423817 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(3,4-dimethoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423818 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(3,5-dimethoxyphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423819 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(benzo[d][1,3]dioxol-5-ylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423820 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-5-(6-(4-(2-(4-tert-butylphenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-N-ethyl-3,4-dihydroxy-tetrahydrofuran-2-carboxamide 44423821 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-(4-morpholinophenylamino)-2-oxoethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 44423822 BindingDB
ADORA2A HGNC:263 P29274 (2S,3S,4R,5R)-N-ethyl-3,4-dihydroxy-5-(6-(4-(2-oxo-2-(pyridin-4-ylamino)ethoxy)phenylamino)-9H-purin-9-yl)-tetrahydrofuran-2-carboxamide 44423823 BindingDB