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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
ADORA2A HGNC:263 P29274 1-(6-(p-toluidino)-9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 44430239 BindingDB
ADORA2A HGNC:263 P29274 1-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-6-(quinolin-2-ylamino)-9H-purin-2-yl)-N-ethyl-1H-pyrazole-4-carboxamide 44430241 BindingDB
ADORA2A HGNC:263 P29274 (R)-tert-butyl 3-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-6-ylamino)pyrrolidine-1-carboxylate 44435354 BindingDB
ADORA2A HGNC:263 P29274 1-((R)-3-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-6-ylamino)pyrrolidin-1-yl)ethanone 44435355 BindingDB
ADORA2A HGNC:263 P29274 (R)-benzyl 3-(9-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)-tetrahydrofuran-2-yl)-9H-purin-6-ylamino)pyrrolidine-1-carboxylate 44435356 BindingDB
ADORA2A HGNC:263 P29274 (1S,2R,4S)-2-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-7-aza-bicyclo[2.2.1]heptane-7-carboxylic acid benzyl ester 44435359 BindingDB
ADORA2A HGNC:263 P29274 (1S,2R,4S)-2-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-7-aza-bicyclo[2.2.1]heptane-7-carboxylic acid 2-chloro-benzyl ester 44435360 BindingDB
ADORA2A HGNC:263 P29274 (1S,2R,4S)-2-[9-((2R,3R,4S,5R)-3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-9H-purin-6-ylamino]-7-aza-bicyclo[2.2.1]heptane-7-carboxylic acid 2-bromo-benzyl ester 44435361 BindingDB
ADORA2A HGNC:263 P29274 8-(Furan-2-yl)-3-[2-(4-phenylpiperazin-1-yl)ethyl]-[1,2,4]triazolo[5,1-f]purin-5-amine 44438076 BindingDB
ADORA2A HGNC:263 P29274 3-Benzyl-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438077 BindingDB
ADORA2A HGNC:263 P29274 3-[(2-Chlorophenyl)methyl]-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438079 BindingDB
ADORA2A HGNC:263 P29274 8-(Furan-2-yl)-3-[2-[4-(4-methoxyphenyl)piperazin-1-yl]ethyl]-[1,2,4]triazolo[5,1-f]purin-5-amine 44438081 BindingDB
ADORA2A HGNC:263 P29274 8-(Furan-2-yl)-3-[2-[4-[4-(2-methoxyethoxy)-2-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]-[1,2,4]triazolo[5,1-f]purin-5-amine 44438082 BindingDB
ADORA2A HGNC:263 P29274 3-[2-[4-(4-Fluorophenyl)piperidin-1-yl]ethyl]-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438083 BindingDB
ADORA2A HGNC:263 P29274 3-[2-[4-(4-Chloro-2-fluorophenyl)piperazin-1-yl]ethyl]-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438084 BindingDB
ADORA2A HGNC:263 P29274 3-[2-[4-(3-Chlorophenyl)piperazin-1-yl]ethyl]-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438085 BindingDB
ADORA2A HGNC:263 P29274 8-(Furan-2-yl)-3-[2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethyl]-[1,2,4]triazolo[5,1-f]purin-5-amine 44438086 BindingDB
ADORA2A HGNC:263 P29274 3-[2-[4-(5-Chloropyridin-2-yl)piperazin-1-yl]ethyl]-8-(furan-2-yl)-[1,2,4]triazolo[5,1-f]purin-5-amine 44438087 BindingDB
ADORA2A HGNC:263 P29274 3-[2-[4-[4-(2-Methoxyethoxy)phenyl]piperazin-1-yl]ethyl]-8-[2-(trifluoromethyl)phenyl]-[1,2,4]triazolo[5,1-f]purin-5-amine 44438091 BindingDB
ADORA2A HGNC:263 P29274 4-[4-[2-[7-Amino-4-(furan-2-yl)-3,5,6,8,10,11-hexazatricyclo[7.3.0.02,6]dodeca-1(9),2,4,7,11-pentaen-10-yl]ethyl]piperazin-1-yl]phenol 44439732 BindingDB