| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TMPRSS2 |
HGNC:11876 |
O15393 |
1-[2-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,4-dimethoxyphenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]ethyl]-3-methylurea |
90666144 |
ChemBL |
| TMPRSS2 |
HGNC:11876 |
O15393 |
1-[2-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,4-dichlorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]ethyl]-3-methylurea |
90666145 |
ChemBL |
| TMPRSS2 |
HGNC:11876 |
O15393 |
1-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,4-dichlorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-3-cyclohexylurea |
90666147 |
ChemBL |
| TMPRSS2 |
HGNC:11876 |
O15393 |
Ms-QFR-Kbt |
135169285 |
GtoPDB |
| TMPRSS2 |
HGNC:11876 |
O15393 |
3-[(2R)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(4,6-dichlorocyclohexa-1,5-dien-1-yl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide |
146025595 |
GtoPDB |
| TMPRSS2 |
HGNC:11876 |
O15393 |
MM3122 |
155925845 |
DrugBank, GtoPDB |
| TMPRSS2 |
HGNC:11876 |
O15393 |
N-(2-carbamimidoyl-3,4-dihydro-1H-isoquinolin-6-yl)naphthalene-2-carboxamide |
171343779 |
ChemBL |
| TMPRSS2 |
HGNC:11876 |
O15393 |
N-(2-carbamimidoyl-3,4-dihydro-1H-isoquinolin-6-yl)-4-methoxybenzamide |
171344680 |
ChemBL |
| TMPRSS2 |
HGNC:11876 |
O15393 |
N-(2-carbamimidoyl-3,4-dihydro-1H-isoquinolin-6-yl)naphthalene-1-carboxamide |
171345025 |
ChemBL |
| TMPRSS4 |
HGNC:11878 |
Q9NRS4 |
5-chloro-2-hydroxy-N-[4-methyl-3,5-bis(trifluoromethyl)phenyl]benzamide |
71508779 |
ChemBL |
| TMPRSS4 |
HGNC:11878 |
Q9NRS4 |
N-[4-bromo-3,5-bis(trifluoromethyl)phenyl]-5-chloro-2-hydroxybenzamide |
71555038 |
ChemBL |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
Leupeptin |
72429 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
4-[4-(4-Carbamimidoylphenyl)piperazin-1-yl]benzenecarboximidamide |
480183 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
4-[4-(4-Carbamimidoylphenyl)-1,4-diazepan-1-yl]benzamidine |
480185 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
alpha,alpha'-Di(amidinophenoxy)-p-xylene |
3000497 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
4-[[2-[(4-Carbamimidoylphenoxy)methyl]phenyl]methoxy]benzamidine |
3010932 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
(2s)-1-[(2r)-2-(Benzylsulfonylamino)-5-Guanidino-Pentanoyl]-N-[(4-Carbamimidoylphenyl)methyl]pyrrolidine-2-Carboxamide |
46899577 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
N-(Benzylsulfonyl)-3-Cyclohexyl-D-Alanyl-N-(4-Carbamimidoylbenzyl)-L-Prolinamide |
46899736 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
3-[(2s)-3-[4-(2-Aminoethyl)piperidin-1-Yl]-2-{[(2',4'-Dichlorobiphenyl-3-Yl)sulfonyl]amino}-3-Oxopropyl]benzenecarboximidamide |
50939649 |
TTD |
| TMPRSS6 |
HGNC:16517 |
Q8IU80 |
3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(2-fluorophenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide |
50939651 |
TTD |