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Drugs And Genes
DRUGs and GENEs
GENE_SYMBOL HGNC_ID UNIPROT_ID DRUG_NAME PUBCHEM_CID Datasource
TMPRSS6 HGNC:16517 Q8IU80 inhibitor 1 [Colombo et al., 2012] 70689167 GtoPDB, TTD
TMPRSS6 HGNC:16517 Q8IU80 Tert-butyl 4-[3-[(3-carbamimidoylphenyl)sulfonylamino]propanoylamino]benzoate;2,2,2-trifluoroacetic acid 71477382 TTD
TMPRSS6 HGNC:16517 Q8IU80 N-[(4-carbamimidoylphenyl)methyl]-3-[(3-carbamimidoylphenyl)sulfonylamino]propanamide;2,2,2-trifluoroacetic acid 71477981 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,4-dichlorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495381 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(2-chloro-4-ethoxyphenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495466 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,3-dichlorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495467 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2-fluorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495468 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(3-fluorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495559 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(3-fluorophenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495560 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(4-fluorophenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495561 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(2,4-dimethoxyphenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495659 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(2,4-dimethoxyphenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495660 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(2,3-dichlorophenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495661 TTD
TMPRSS6 HGNC:16517 Q8IU80 4-[1-[(2S)-3-(3-carbamimidoylphenyl)-2-[[3-(3,4-dichlorophenyl)phenyl]sulfonylamino]propanoyl]piperidin-4-yl]-N-methylbutanamide 71495765 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[[3-(3,4-dichlorophenyl)phenyl]sulfonylamino]-3-oxopropyl]benzenecarboximidamide 71495766 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-amino-N-[3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-[2-(carbamoylamino)ethyl]piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl]propanamide 71495974 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-amino-N-[3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-(methylcarbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl]propanamide 71495975 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-amino-N-[3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-(carbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl]propanamide 71495976 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-amino-N-[3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-(ethylcarbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl]propanamide 71495977 TTD
TMPRSS6 HGNC:16517 Q8IU80 3-amino-N-[3-[[(2S)-3-(3-carbamimidoylphenyl)-1-[4-(cyclohexylcarbamoylamino)piperidin-1-yl]-1-oxopropan-2-yl]sulfamoyl]phenyl]propanamide 71496089 TTD