| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
Unii-DQ4lkh74UY |
16742146 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-(propan-2-yl)phenyl}methyl)-3-1H-indazol-4-ylurea |
16747867 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-(3,3-dimethylbutyl)phenyl}methyl)-3-1H-indazol-4-ylurea |
16747868 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-{[4-(Azepan-1-yl)-2-chlorophenyl]methyl}-1-isoquinolin-5-ylurea |
16748125 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-{[4-(Azepan-1-yl)-3-(trifluoromethyl)phenyl]methyl}-1-isoquinolin-5-ylurea |
16748127 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-{[4-(2,3-dihydro-1H-isoindol-2-yl)-3-fluorophenyl]methyl}-1-(3-methylisoquinolin-5-yl)urea |
16748248 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-{[4-(azepan-1-yl)-2-(trifluoromethyl)phenyl]methyl}-3-1H-indazol-4-ylurea |
16748249 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]phenyl}methyl)-3-1H-indazol-4-ylurea |
16748250 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-(trifluoromethyl)phenyl}methyl)-3-1H-indazol-4-ylurea |
16748251 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-bromophenyl}methyl)-3-1H-indazol-4-ylurea |
16748252 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3,5-difluorophenyl}methyl)-3-1H-indazol-4-ylurea |
16748373 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2,5-difluorophenyl}methyl)-3-1H-indazol-4-ylurea |
16748374 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-{4-[6-(4-Trifluoromethyl-cyclohex-1-enyl)-pyrimidin-4-yloxy]-benzothiazol-2-yl}-acetamide |
16748464 |
ChemBL |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-Isoquinolin-5-yl-3-{[4-(piperidin-1-yl)phenyl]methyl}urea |
16749133 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-Isoquinolin-5-yl-3-{[4-(4-methylpiperidin-1-yl)phenyl]methyl}urea |
16749136 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]phenyl}methyl)-1-isoquinolin-5-ylurea |
16749139 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-{[4-(Azepan-1-yl)-2-(trifluoromethyl)phenyl]methyl}-1-isoquinolin-5-ylurea |
16749240 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(3-aminoisoquinolin-5-yl)-3-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-(trifluoromethyl)phenyl}methyl)urea |
16749243 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-{[4-(azepan-1-yl)-2-chlorophenyl]methyl}-3-1H-indazol-4-ylurea |
16749244 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-{[4-(azepan-1-yl)-3-(trifluoromethyl)phenyl]methyl}-3-1H-indazol-4-ylurea |
16749350 |
ChemBL, TTD |