| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-{[4-(azepan-1-yl)-3,5-difluorophenyl]methyl}-3-1H-indazol-4-ylurea |
16749351 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-chlorophenyl}methyl)-3-1H-indazol-4-ylurea |
16749352 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-(trifluoromethyl)phenyl}methyl)-3-1H-indazol-4-ylurea |
16749353 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-chlorophenyl}methyl)-3-1H-indazol-4-ylurea |
16749354 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-fluorophenyl}methyl)-3-1H-indazol-4-ylurea |
16749355 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[6-(4-tert-butylphenyl)pyrimidin-4-yl]quinolin-7-amine |
16749438 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2,3-difluorophenyl}methyl)-3-1H-indazol-4-ylurea |
16749462 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1S,5R)-8-azaspiro[bicyclo[3.2.1]octane-3,2''-[1,3]dioxolane]]-2,5-difluorophenyl}methyl)-3-1H-indazol-4-ylurea |
16749463 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({2,5-difluoro-4-[(1R,5S)-3-oxo-8-azabicyclo[3.2.1]octan-8-yl]phenyl}methyl)-3-1H-indazol-4-ylurea |
16749464 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-(1-methyl-1H-indazol-4-yl)-1-[(1-methyl-1H-indol-5-yl)methyl]urea |
16749465 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-1H-indazol-4-ylurea |
16749466 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-[(1-ethyl-2,3-dihydro-1H-indol-5-yl)methyl]-3-(1-methyl-1H-indazol-4-yl)urea |
16749467 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
3-1H-indazol-4-yl-1-[(9-methyl-9H-carbazol-3-yl)methyl]urea |
16749565 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-3-methylphenyl}methyl)-3-1H-indazol-4-ylurea |
16749566 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-methylphenyl}methyl)-3-1H-indazol-4-ylurea |
16749567 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-(2-benzyl-4-(8-azabicyclo[3.2.1]octan-8-yl)benzyl)-3-(1H-indazol-4-yl)urea |
16749568 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-({4-[(1R,5S)-8-azabicyclo[3.2.1]octan-8-yl]-2-benzylphenyl}methyl)-3-(1-methyl-1H-indazol-4-yl)urea |
16749569 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
N-[2-(5-methoxy-1H-indol-3-yl)ethyl]-4-(trifluoromethyl)benzamide |
17026579 |
ChemBL, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
Mavatrep |
17751090 |
ChemBL, GtoPDB, Pubchem, TTD |
| TRPV1 |
HGNC:12716 |
Q8NER1 |
1-[(1R)-5-tert-butyl-2,3-dihydro-1H-inden-1-yl]-3-isoquinolin-5-ylurea |
17757384 |
ChemBL, GtoPDB |