| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Gsk-1059615 |
23582824 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
3-(2-(1-(2-(dimethylamino)acetyl)-6-methoxy-1,2,3,4-tetrahydroquinolin-7-ylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)thiophene-2-carboxamide |
25210971 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
3-[(2-{[1-(N,N-Dimethylglycyl)-6-Methoxy-4,4-Dimethyl-1,2,3,4-Tetrahydroquinolin-7-Yl]amino}-7h-Pyrrolo[2,3-D]pyrimidin-4-Yl)amino]thiophene-2-Carboxamide |
25210972 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
2-((2-((5-(2-(Dimethylamino)acetamido)-2-methoxy-4-methylphenyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-6-fluorobenzamide |
25211574 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
4-Fluoro-2-((2-((2-methoxy-4-(1-propylpiperidin-3-yl)phenyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)benzamide |
25218600 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
4-fluoro-2-[(2-{[2-methoxy-4-(1-propylpiperidin-4-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide |
25218601 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
5-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide |
25218614 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
N-(2-(2-(2-Methoxy-4-morpholinophenylamino)-5-fluoropyrimidin-4-ylamino)phenyl)methanesulfonamide |
44252884 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Azd-4547 |
51039095 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
3-[[2-[[1-[2-(dimethylamino)acetyl]-6-methoxy-3,4-dihydro-2H-quinolin-7-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]-N-methylpyridine-2-carboxamide |
53239988 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
7-methyl-5-(1-((3-(trifluoromethyl)phenyl)acetyl)-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo(2,3-d)pyrimidin-4-amine |
53469448 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-[(1R)-2-amino-1-phenylethoxy]-1-ethylimidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol;2,2,2-trifluoroacetic acid |
56604034 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
5-Chloro-4-(1H-indol-3-yl)-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidin-2-amine |
56655374 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Ceritinib |
57379345 |
ChemBL, GtoPDB, Pubchem |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
4-[6-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide |
59603829 |
ChemBL |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
2-anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one |
69036886 |
ChemBL |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Otssp167 |
135398499 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Dovitinib |
135398510 |
DGidb |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
(5Z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5H)-one |
135400873 |
DSigDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
Nintedanib |
135423438 |
Pubchem |