| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
4-({5-chloro-4-[(cis-4-hydroxy-4-methylcyclohexyl)oxy]-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)-N,N-dimethyl-3-{[(2R)-1,1,1-trifluoropropan-2-yl]oxy}benzamide |
138320062 |
ChemBL, GtoPDB |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide |
155531579 |
ChemBL |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide |
155552127 |
ChemBL |
| TSSK1B |
HGNC:14968 |
Q9BXA7 |
TTK inhibitor 3 |
162640906 |
ChemBL |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
Staurosporine |
44259 |
ChemBL, TTD |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
Alsterpaullone |
5005498 |
DGidb |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
5-(5,6-Dimethoxybenzimidazol-1-yl)-3-[[2-(trifluoromethyl)phenyl]methoxy]thiophene-2-carboxamide |
9826308 |
DGidb |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
Cenisertib |
11569967 |
DGidb |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
5-chloro-N4-(2-(isopropylsulfonyl)phenyl)-N2-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidine-2,4-diamine |
16038120 |
DGidb |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
2-(6-Methoxy-1-Oxo-1,3-Dihydro-2h-Isoindol-2-Yl)-N-[4-(Piperazin-1-Yl)pyridin-3-Yl]-1,3-Thiazole-4-Carboxamide |
24951610 |
ChemBL, TTD |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
3-(2-(1-(2-(dimethylamino)acetyl)-6-methoxy-1,2,3,4-tetrahydroquinolin-7-ylamino)-7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)thiophene-2-carboxamide |
25210971 |
DSigDB |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
3-[(2-{[1-(N,N-Dimethylglycyl)-6-Methoxy-4,4-Dimethyl-1,2,3,4-Tetrahydroquinolin-7-Yl]amino}-7h-Pyrrolo[2,3-D]pyrimidin-4-Yl)amino]thiophene-2-Carboxamide |
25210972 |
DSigDB |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
4-Fluoro-2-((2-((2-methoxy-4-(1-propylpiperidin-3-yl)phenyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)benzamide |
25218600 |
DSigDB |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
4-fluoro-2-[(2-{[2-methoxy-4-(1-propylpiperidin-4-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide |
25218601 |
DSigDB |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
5-fluoro-2-{[2-({2-methoxy-4-[4-(propan-2-yl)piperazin-1-yl]phenyl}amino)-7H-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide |
25218614 |
DSigDB |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
N-[(1S)-1-(5-fluoropyridin-2-yl)ethyl]-3-(3-propan-2-yloxy-1H-pyrazol-5-yl)imidazo[4,5-b]pyridin-5-amine |
59627005 |
GtoPDB, TTD |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
Rg-1530 |
135398512 |
DGidb |
| TSSK2 |
HGNC:11401 |
Q96PF2 |
TTK inhibitor 3 |
162640906 |
ChemBL |
| TSSK3 |
HGNC:15473 |
Q96PN8 |
Staurosporine |
44259 |
ChemBL |
| TSSK3 |
HGNC:15473 |
Q96PN8 |
Ceritinib |
57379345 |
DSigDB |