| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-(4-(1,2-dimethyl-1H-imidazol-5-yl)-2-methoxyphenyl)-8-(1-methyl-1H-pyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386771 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
tert-butyl 4-(4-(3-((2-methoxy-4-(3-methoxyazetidine-1-carbonyl)phenyl)-amino)isoquinolin-5-yl)-1H-pyrazol-1-yl)piperidine-1-carboxylate |
73386772 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxy-4-((5-(1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl)isoquinolin-3-yl)amino)phenyl)(3-methoxyazetidin-1-yl)methanone |
73386773 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxy-4-((5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)isoquinolin-3-yl)amino)phenyl)(3-methoxyazetidin-1-yl)methanone |
73386774 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[5-[1-[2-(Dimethylamino)ethyl]pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
73386775 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(cyclopropylmethoxy)-N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
73386776 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
1-[[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]-2-methylpropan-2-ol |
73386777 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(2-methoxy-6-morpholinopyridin-3-yl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
73386778 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(2-methoxy-6-(methylsulfonyl)pyridin-3-yl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
73386779 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(2-methoxy-4-(1-methyl-1H-imidazol-5-yl)phenyl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
73386780 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-methoxyphenyl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
73386781 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-(1,5-dimethylpyrazol-4-yl)-2-methoxyphenyl]-8-N-[(3-methyloxolan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
73386782 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(2-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386783 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(4-chloro-2-methoxyphenyl)-8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386785 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2,4-dichlorophenyl)-8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386786 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-Methoxy-2-[[2-[2-methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]propan-1-ol |
73386787 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-chloro-N,N-dimethyl-4-[[5-(1-methylpyrazol-4-yl)isoquinolin-3-yl]amino]benzamide |
73386864 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-methoxy-N,N-dimethyl-4-[[5-(1-methylpyrazol-4-yl)isoquinolin-3-yl]amino]benzamide |
73386865 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[5-(1-methylpyrazol-4-yl)isoquinolin-3-yl]amino]phenyl]methanone |
73386866 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-chloro-4-(1-methylpyrazol-4-yl)phenyl]-5-(1-methylpyrazol-4-yl)isoquinolin-3-amine |
73386867 |
ChemBL |