| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
73386891 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-8-N-[(3-methyloxolan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
73386892 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-cyclopropyl-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidin-2-amine |
73386970 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-5-methyl-4-(1-methylpyrazol-4-yl)phenyl]-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386971 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
(3-Methoxyazetidin-1-yl)-[3-methoxy-4-[[5-(2-methylpyrazol-3-yl)isoquinolin-3-yl]amino]phenyl]methanone |
73386972 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[5-(1,3-Dimethylpyrazol-4-yl)isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
73386973 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[5-(3,5-Dimethyl-1,2-oxazol-4-yl)isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
73386975 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(1-methyl-1H-pyrazol-4-yl)-N-(2-methyl-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
73386976 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(4-methylpiperazin-1-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386977 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(3,3-difluoroazetidin-1-yl)-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidin-2-amine |
73386978 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(1-propan-2-ylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386979 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(1-ethyl-1H-pyrazol-4-yl)-N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
73386980 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(3-methoxyazetidin-1-yl)-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidin-2-amine |
73386981 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-[1-(2,2-difluoroethyl)pyrazol-4-yl]-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidin-2-amine |
73386982 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(3-methoxy-2,2-dimethylpropyl)-2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
73386983 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2-methoxy-2-methylpropyl)-2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
73386984 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-(2,2,2-trifluoroethyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
73386985 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-amine |
73386986 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2,2-dimethylpropyl)-2-N-(2-methoxy-4-piperidin-1-ylphenyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
73386987 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-(3,6-Dihydro-2H-pyran-4-yl)-N-(2-methoxy-4-(1-methyl-1H-pyrazol-4-yl)phenyl)pyrido[3,4-d]pyrimidin-2-amine |
73386988 |
ChemBL |