| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
2-N-[6-(2,3-dimethylimidazol-4-yl)-2-methoxypyridin-3-yl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90000927 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-(difluoromethoxy)-4-(1-methylpyrazol-4-yl)phenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90000930 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N2-(4-(1,5-dimethyl-1H-pyrazol-4-yl)-2-methoxyphenyl)-N8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine |
90000938 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-(1,5-dimethylpyrazol-4-yl)-2-methoxyphenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90000975 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-methoxy-4-[[8-[(2-methoxy-2-methylpropyl)amino]pyrido[3,4-d]pyrimidin-2-yl]amino]-N,N-dimethylbenzamide |
90000976 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2-methoxy-2-methylpropyl)-2-N-[2-methoxy-4-(1-methyltetrazol-5-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
90000987 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-[3-(2-methoxyethyl)-2-methylimidazol-4-yl]phenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90000997 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[5-[3-Methoxy-4-[[6-[1-(2-methoxyethyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]-1-methylimidazol-2-yl]methanol |
90001012 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-(1,3-dimethylpyrazol-4-yl)-2-methoxyphenyl]-8-N-[(3-methyloxolan-3-yl)methyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
90001016 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[3-Methoxy-4-[[8-[(2-methoxy-2-methylpropyl)amino]pyrido[3,4-d]pyrimidin-2-yl]amino]phenyl]-(4-methylpiperazin-1-yl)methanone |
90001028 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-[[2-[2-Methoxy-4-(1-methylpyrazol-4-yl)anilino]pyrido[3,4-d]pyrimidin-8-yl]amino]propane-1,3-diol |
90001044 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-chloro-2-(difluoromethoxy)phenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90001045 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[6-(1,5-dimethylpyrazol-4-yl)-2-methoxypyridin-3-yl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90001055 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-(oxolan-3-ylmethyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90001094 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(3-Hydroxy-3-methylbutan-2-yl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
90001100 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2,2-dimethylpropyl)-2-N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine |
90001169 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2-methoxy-2-methylpropyl)-2-N-[2-methoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-6-methylpyrido[3,4-d]pyrimidine-2,8-diamine |
90001170 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-N-methylpyrido[3,4-d]pyrimidine-2,8-diamine |
90001192 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-Chloro-4-[[8-(2-oxa-7-azaspiro[3.4]octan-7-yl)pyrido[3,4-d]pyrimidin-2-yl]amino]benzonitrile |
90001273 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[4-(1-ethylpyrazol-4-yl)-2-methoxyphenyl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
90001325 |
ChemBL |