| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[7-[(4-hydroxycyclohexyl)methylamino]-5-pyridin-3-yloxypyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
90176191 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-Cyclopropyl-2-Methyl-4-(7-{[2-(Morpholin-4-Yl)ethyl]amino}-5-Phenoxypyrazolo[1,5-A]pyrimidin-3-Yl)benzamide |
90176196 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[5-(cyclopentylamino)-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-N-cyclopropyl-2-methylbenzamide |
90176199 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[2-(cyclopentylamino)-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-N-cyclopropyl-2-fluorobenzamide |
90176200 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[2-anilino-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-N-cyclopropyl-2-methylbenzamide |
90176227 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-{2-Methoxy-4-[(1-Methylpiperidin-4-Yl)oxy]phenyl}-4-(1h-Pyrrolo[2,3-C]pyridin-3-Yl)pyrimidin-2-Amine |
91668530 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
Mps1-IN-3 |
91885443 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
Jak3-IN-1 |
92042864 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-(dimethylamino)-2-phenyl-N-[3-(3-sulfamoylphenyl)-1H-indazol-5-yl]acetamide |
101902997 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-phenyl-2-pyrrolidin-1-yl-N-[3-(3-sulfamoylphenyl)-1H-indazol-5-yl]acetamide |
101902998 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-pyrrolidin-1-yl-N-[3-(3-sulfamoylphenyl)-1H-indazol-5-yl]-2-thiophen-3-ylacetamide |
101902999 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[3-(Aminosulfonyl)phenyl]-1H-indazole-5-yl]-2-(dimethylamino)-2-(2-ethylphenyl)acetamide |
101903000 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[6-(2-fluoro-4-hydroxyphenoxy)-4-(3,3,3-trifluoropropylamino)benzimidazol-1-yl]-N,2-dimethylbenzamide |
117628699 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-ethyl-4-[6-(3-hydroxyphenoxy)-4-(3,3,3-trifluoropropylamino)benzimidazol-1-yl]-2-methylbenzamide |
117629252 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[6-(4-methoxy-2-methylsulfanylphenoxy)-4-(oxan-4-ylmethylamino)benzimidazol-1-yl]-2-methylbenzamide |
117629306 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-2-methyl-4-[6-phenoxy-4-(3,3,3-trifluoropropylamino)benzimidazol-1-yl]benzamide |
117634689 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[cyclobutyl(thiophen-3-yl)methyl]-3-[4-[[(1S,5R)-8-formyl-8-azabicyclo[3.2.1]octan-3-yl]oxy]phenyl]-1H-indazole-5-carboxamide |
117737852 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(1-morpholin-4-ylcyclohexyl)methyl]-3-(4-morpholin-4-ylphenyl)-1H-indazole-5-carboxamide |
117738442 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-[4-(4-methylpiperazin-1-yl)phenyl]-N-[(1-morpholin-4-ylcyclohexyl)methyl]-1H-indazole-5-carboxamide |
117738670 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US9663510, Example comparitive example 4 |
117749351 |
ChemBL |