| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-[(S)-cyclopropyl-(2-fluorophenyl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751252 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(R)-cyclopropyl-(2-fluorophenyl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751256 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[(S)-cyclopropyl(pyridin-2-yl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751333 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(1S)-1-(2-chlorophenyl)-2-methylpropyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751334 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[(S)-cyclopentyl(pyridin-2-yl)methyl]-3-[4-(3-oxa-9-azabicyclo[3.3.1]nonan-9-yl)phenyl]-1H-indazole-5-carboxamide |
117751336 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(R)-cyclopentyl(pyridin-2-yl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751337 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[(R)-cyclopropyl(pyridin-2-yl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751339 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[(1-morpholin-4-ylcyclohexyl)methyl]-3-[4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)phenyl]-1H-indazole-5-carboxamide |
117751349 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(1-morpholin-4-ylcyclohexyl)methyl]-3-[4-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)phenyl]-1H-indazole-5-carboxamide |
117751357 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
4-((4-(Cyclopentyloxy)-5-(2-methylbenzo[d]oxazol-6-yl)-7H-pyrrolo-[2,3-d]pyrimidin-2-yl)amino)-3-methoxy-N-methylbenzamide |
117881270 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[7-[(3-hydroxy-3-methylcyclobutyl)methylamino]-5-pyridin-3-yloxypyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118086034 |
ChemBL, GtoPDB, Pubchem, TTD |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
118274570 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[1-(2-Hydroxy-2-methylpropyl)triazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
118274574 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[2-[1-(2-Hydroxy-2-methylpropyl)pyrazol-4-yl]-1,6-naphthyridin-7-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
118274581 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[5-[3-Methoxy-4-[[6-[1-(2-methoxyethyl)pyrazol-4-yl]isoquinolin-3-yl]amino]phenyl]-2-methylimidazol-1-yl]methanol |
118283448 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
[4-[[6-[2-(2-Hydroxy-2-methylpropyl)triazol-4-yl]isoquinolin-3-yl]amino]-3-methoxyphenyl]-(3-methoxyazetidin-1-yl)methanone |
118283450 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-6-(3-methylimidazol-4-yl)pyridin-3-yl]-8-N-(2-methoxy-2-methylpropyl)pyrido[3,4-d]pyrimidine-2,8-diamine |
118331539 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-N-(2-methoxy-2-methylpropyl)-2-N-[2-methoxy-4-(2-methyl-1,2,4-triazol-3-yl)phenyl]-6-methylpyrido[3,4-d]pyrimidine-2,8-diamine |
118331597 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 4 |
118348977 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 56 |
118348985 |
ChemBL, TTD |