| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
8-(3,3-dimethylazetidin-1-yl)-N-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-6-methylpyrido[3,4-d]pyrimidin-2-amine |
118349012 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 7 |
118349055 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-(3-fluorophenoxy)-7-(2-morpholin-4-ylethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118452766 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[2-(cyclopentylamino)-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-N-cyclopropylbenzamide |
118452767 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[4-(oxan-4-ylmethylamino)-2-phenoxypyrazolo[1,5-a][1,3,5]triazin-8-yl]benzamide |
118452789 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-[[(1S,2R)-2-hydroxycyclohexyl]amino]-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118452843 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-[[(1S)-1-cyclopropyl-2-hydroxy-2-methylpropyl]amino]-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118452846 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-[[(2R)-1-hydroxybutan-2-yl]amino]-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118452870 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[2-(2,3-difluorophenoxy)-4-(2-morpholin-4-ylethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-2-methylbenzamide |
118458718 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-[[(1R,2R)-2-hydroxycyclohexyl]amino]-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118458775 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[7-[(3-hydroxycyclobutyl)methylamino]-5-pyridin-3-yloxypyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
118458786 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[[[5-chloro-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
118475621 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[[[5-chloro-2-[[1-(2-hydroxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
118475644 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[[[5-chloro-2-(3,5-difluoro-4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
118475649 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[[[5-chloro-2-[[1-(2-methoxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
118475652 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-[3-[[[5-chloro-2-(4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
118475705 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[6-ethynyl-8-(3,3,3-trifluoropropylamino)imidazo[1,2-a]pyrazin-3-yl]-N-[(2S)-2-fluorocyclopropyl]-2-methylbenzamide |
118543779 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-(4-chloro-1H-indazol-3-yl)benzenesulfonamide |
118712905 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
3-[4-(2,6-difluorophenyl)-1H-indazol-3-yl]benzenesulfonamide |
118712909 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
3-(6-phenyl-1H-indazol-3-yl)benzenesulfonamide |
118712910 |
ChemBL, TTD |