| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-[(1R)-2-cyclopropyl-1-pyridin-2-ylethyl]-3-[4-[(1S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]phenyl]-1H-indazole-5-carboxamide |
118735397 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-[4-[(1S,5S)-3-hydroxy-9-azabicyclo[3.3.1]nonan-9-yl]phenyl]-N-[(1S)-3-methyl-1-pyridin-2-ylbutyl]-1H-indazole-5-carboxamide |
118735398 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
3-[4-[(1R,5R)-7-hydroxy-3-oxa-9-azabicyclo[3.3.1]nonan-9-yl]phenyl]-N-[(1S)-3-methyl-1-pyridin-2-ylbutyl]-1H-indazole-5-carboxamide |
118735399 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-[(R)-cyclopentyl(pyridin-2-yl)methyl]-3-[4-[(1R,5R)-7-hydroxy-3-oxa-9-azabicyclo[3.3.1]nonan-9-yl]phenyl]-1H-indazole-5-carboxamide |
118735400 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
4-[6-(cyclohexylamino)-8-[(2-hydroxy-2-methylpropyl)amino]imidazo[1,2-b]pyridazin-3-yl]-N-cyclopropylbenzamide |
118735401 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-(Furan-3-Yl)-3-Phenyl-2~{h}-Pyrazolo[4,3-C]pyridine |
119025602 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-(2,4-dimethoxyphenyl)-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
119025603 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-N-(2-methoxyphenyl)-4-N-(2-propan-2-ylsulfonylphenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
121320413 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-N-cyclohexyl-2-N-(2-methoxy-4-morpholin-4-ylphenyl)-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamine |
121320416 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-[8-(3-aminopropylamino)-3-[4-(2-cyclopropyl-1H-imidazol-5-yl)phenyl]imidazo[1,2-a]pyrazin-6-yl]ethynol |
122164745 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
5-[3-[4-(Cyclopropylcarbamoyl)phenyl]-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-6-yl]pent-4-ynoic acid |
122164746 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
4-[6-(4-cyclohexylbut-1-ynyl)-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]-N-cyclopropylbenzamide |
122164747 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[6-[(3R)-3-hydroxyoct-1-ynyl]-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide |
122164748 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
Methyl 5-[3-[4-(cyclopropylcarbamoyl)phenyl]-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-6-yl]pent-4-ynoate |
122164749 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
8-[3-[4-(Cyclopropylcarbamoyl)phenyl]-8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-6-yl]oct-7-ynoic acid |
122164750 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(2,6-diethylphenyl)-2-[2-methoxy-4-(4-methylpiperazin-1-yl)anilino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide |
122632882 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 54 |
124124034 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 3 |
124124085 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
US10399974, Example 42 |
124124180 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
(2S)-2-(4-fluorophenyl)-N-[4-[2-(2-methoxy-4-methylsulfonylanilino)-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamide |
124672819 |
ChemBL |