| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-(phenylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide |
126473390 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-(4-methoxyphenyl)-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine |
127044233 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
2-chloro-N-cyclopropyl-4-[2-(oxan-4-ylamino)-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]benzamide |
127048362 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[2-(3-fluoroanilino)-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-2-methylbenzamide |
127049041 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[2-(2-fluoroanilino)-4-(oxan-4-ylmethylamino)pyrazolo[1,5-a][1,3,5]triazin-8-yl]-2-methylbenzamide |
127052461 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
4-[[5-(1,3-dimethylpyrazol-4-yl)isoquinolin-3-yl]amino]-N-(1-methylpiperidin-4-yl)-3-(trifluoromethoxy)benzamide |
129625762 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-3-[[(3R)-3-methyloxolan-3-yl]methyl]-4H-pyrido[3,4-d]pyrimidine-2,8-diamine |
129625763 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
2-N-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-3-[[(3S)-3-methyloxolan-3-yl]methyl]-4H-pyrido[3,4-d]pyrimidine-2,8-diamine |
129625764 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[7-[(3-hydroxy-3-methylcyclobutyl)methylamino]-5-pyridin-2-yloxypyrazolo[1,5-a]pyridin-3-yl]-2-methylbenzamide |
129626596 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[5-[[(1S,2R)-2-hydroxycyclopentyl]amino]-7-(oxan-4-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzamide |
130289079 |
ChemBL, TTD |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(R)-methylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635843 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(R)-ethylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635844 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[6-phenyl-8-[(R)-propylsulfinyl]imidazo[1,2-a]pyrazin-3-yl]benzamide |
131635845 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
4-[8-[(R)-butylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]-N-cyclopropylbenzamide |
131635846 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(R)-3,3-dimethylbutylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635847 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[[(2R)-oxolan-2-yl]methylsulfanyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635848 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[[(2R)-oxolan-2-yl]methylsulfonyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635849 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(R)-2-methylpropylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635850 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[8-[(R)-3-methylbutylsulfinyl]-6-phenylimidazo[1,2-a]pyrazin-3-yl]benzamide |
131635851 |
ChemBL |
| TTK |
HGNC:12401 |
P33981 |
N-cyclopropyl-4-[6-phenyl-8-[(R)-2,2,2-trifluoroethylsulfinyl]imidazo[1,2-a]pyrazin-3-yl]benzamide |
131635852 |
ChemBL |