| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
Cyclopropanecarboxylic acid [5-(4-methoxy-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]-amide |
24798571 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-phenyl-N-(3,4,5-trimethoxyphenyl)benzo[d]oxazol-2-amine |
24800423 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-(quinolin-6-yl)-N-(3,4,5-trimethoxyphenyl)benzo[d]oxazol-2-amine |
24800776 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-(4-(2-(3,4,5-trimethoxyphenylamino)benzo[d]oxazol-7-yl)phenyl)methanesulfonamide |
24801129 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-(pyridin-2-yl)-N-(3,4,5-trimethoxyphenyl)benzo[d]oxazol-2-amine |
24801650 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-14-methyl-5,7,14,20,29-pentazapentacyclo[18.5.2.12,6.18,12.023,27]nonacosa-1(26),2(29),3,5,8,10,12(28),16,21,23(27),24-undecaene |
24899557 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Momelotinib |
25062766 |
ChemBL, DGidb, DSigDB, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Defactinib |
25117126 |
ChemBL, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Morpholino(4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)phenyl)methanone |
25123154 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-Morpholino-2-(4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)phenyl)ethanone |
25123155 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-(1,1-Dioxo-1,4-thiazinan-4-yl)-2-[4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]phenyl]ethanone |
25123472 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(2-Methyl-4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)phenyl)(morpholino)methanone |
25123475 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
8-[4-(1,1-Dioxo-1lambda*6*-thiomorpholin-4-ylmethyl)-phenyl]-2-(3,4,5-trimethoxy-phenyl)-quinoxaline |
25123806 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-Fluoro-4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)benzyl)morpholine |
25123807 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
8-(3-Methyl-4-morpholin-4-ylmethyl-phenyl)-2-(3,4,5-trimethoxy-phenyl)-quinoxaline |
25123808 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Ruxolitinib |
25126798 |
ChemBL, DGidb, DrugBank, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Ruxolitinib Phosphate |
25127112 |
Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamide |
25128110 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-11-(2-pyrrolidin-1-ylethoxy)-14,20-dioxa-5,7,22,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8(26),9,11,16,21,23-decaene |
25154395 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-3-methyl-11-(2-pyrrolidin-1-ylethoxy)-14,20-dioxa-5,7,22,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8(26),9,11,16,21,23-decaene |
25154436 |
TTD |