| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
N-[(2z)-4-(3-Fluoro-5-Morpholin-4-Ylphenyl)pyrimidin-2(1h)-Ylidene]-4-(3-Morpholin-4-Yl-1h-1,2,4-Triazol-1-Yl)aniline |
25222038 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
N-methyl-6-[[4-(2-propan-2-ylsulfonylanilino)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino]-3-pyridinecarboxamide |
25226483 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
2-chloro-6-fluoro-N-(pyridin-4-yl)benzamide |
25236808 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Foretinib |
42642645 |
Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Baricitinib |
44205240 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Dabrafenib |
44462760 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
1-(6,7-dimethoxyquinazolin-4-yl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-amine |
44551660 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
5-(2-chlorophenyl)-1H-indazol-3-amine |
44570390 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Cerdulatinib |
44595079 |
ChemBL, DGidb, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Solcitinib |
44603362 |
ChemBL, DGidb, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-[4-(morpholin-4-ylmethyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide |
44626045 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Oclacitinib |
44631938 |
ChemBL, DGidb, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
5-amino-N-[5-(2,5-dichlorophenyl)-1H-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
45375833 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-(3-methyl-1,2-oxazol-5-yl)-5-[3-(trifluoromethyl)anilino]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
46191142 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Ilorasertib |
46207586 |
DGidb |
| TYK2 |
HGNC:12440 |
P29597 |
Gandotinib |
46213929 |
ChemBL, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Pacritinib |
46216796 |
ChemBL, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
5-(2-aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amine |
46224684 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2,6-difluoro-4-(3-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)quinoxalin-5-yl)benzyl)morpholine |
46398810 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-Chloro-15-oxa-2,4,8,25-tetrazatetracyclo[17.3.1.13,7.110,14]pentacosa-1(22),3,5,7(25),10(24),11,13,19(23),20-nonaene |
46835839 |
ChemBL |