| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
Morpholino(4-(2-(3,4,5-trimethoxyphenylamino)benzo[d]oxazol-7-yl)phenyl)methanone |
46880687 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(2-Fluoro-4-(2-(3,4,5-trimethoxyphenylamino)benzo[d]oxazol-7-yl)phenyl)(morpholino)methanone |
46880737 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-(4-(morpholinomethyl)phenyl)-N-(3,4,5-trimethoxyphenyl)benzo[d]oxazol-2-amine |
46880738 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N,N-dimethyl-4-(7-(4-(morpholine-4-carbonyl)phenyl)benzo[d]oxazol-2-ylamino)benzamide |
46880739 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(2-Methyl-4-(2-(4-(4-methylpiperazin-1-yl)phenylamino)benzo[d]oxazol-7-yl)phenyl)(morpholino)methanone |
46880784 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(7-(3,5-difluoro-4-(morpholinomethyl)phenyl)benzo[d]oxazol-2-ylamino)-N-(3-(dimethylamino)propyl)-2-methylbenzamide |
46880785 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(3-Methyl-4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)benzyl)morpholine |
46885231 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(3-Fluoro-4-(3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl)benzyl)morpholine |
46885232 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
[4-[8-[4-[(1,1-Dioxo-1,4-thiazinan-4-yl)methyl]phenyl]quinoxalin-2-yl]-2-methylphenyl]-(4-methylpiperazin-1-yl)methanone |
46885233 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(2-Methyl-4-(8-(3-methyl-4-(morpholinomethyl)phenyl)quinoxalin-2-yl)phenyl)(morpholino)methanone |
46885234 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(4-(8-(3-Fluoro-4-(morpholinomethyl)phenyl)quinoxalin-2-yl)-2-methylphenyl)(morpholino)methanone |
46885289 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(4-(8-(3,5-Difluoro-4-(morpholinomethyl)phenyl)quinoxalin-2-yl)-2-methylphenyl)(morpholino)methanone |
46885290 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Ac-430 |
46892373 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
3-(1h-Indol-3-Yl)-4-[2-(4-Oxopiperidin-1-Yl)-5-(Trifluoromethyl)pyrimidin-4-Yl]-1h-Pyrrole-2,5-Dione |
49817363 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Acetamide, N-[2-[6-[[4-(cyclobutylamino)-5-(trifluoromethyl)-2-pyrimidinyl]amino]-1,2,3,4-tetrahydronaphthalen-1,4-imin-9-yl]-2-oxoethyl]- |
49830590 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Filgotinib |
49831257 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-(4-(5-chloro-2-methoxyphenyl)-2-methylthiazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide |
49836036 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1S,2R)-1-N-[4-[(2,6-dichlorobenzoyl)amino]pyridin-2-yl]cyclopropane-1,2-dicarboxamide |
49839198 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2,6-dichloro-N-[2-[(1-ethylpyrazol-4-yl)amino]pyridin-4-yl]benzamide |
49839441 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2,6-Dichloro-N-{2-[(Cyclopropylcarbonyl)amino]pyridin-4-Yl}benzamide |
49839561 |
ChemBL, TTD |