| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
2,6-dichloro-N-[2-(cyclopropanecarbonylamino)pyridin-4-yl]-4-ethynylbenzamide |
49839914 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
8-Cyclohexyl-3h-dipyrrolo[1,2-a:2',3'-e]pyrazine |
49850211 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-(4-cyanopiperidin-1-yl)-1H-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
49855517 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[1-(2-hydroxy-2-methylpropyl)-3-(2-methylpiperidin-1-yl)pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
49855709 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-(5-chloro-2-oxopyridin-1-yl)-1H-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
49856093 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-((3R,4R)-1-benzyl-4-methylpiperidin-3-yl)-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine |
49856703 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-(1-(5-chloro-2-methylphenyl)-3-methyl-1H-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide |
49856844 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-(Cyclopentylamino)pyrrolo[1,2-b]pyridazine-3-carboxamide |
50914031 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Delgocitinib |
50914062 |
ChemBL, DGidb, GtoPDB, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
Bms-911543 |
50922691 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-[5-[4-(2-Hydroxy-2-methyl-1-oxopropyl)-1-piperazinyl]-2-(trifluoromethyl)phenyl]-4-(1H-indol-3-yl)-1H-pyrrole-2,5-dione |
50925411 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-{3-[4-(1H-Indol-3-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-3-yl]-4-trifluoromethyl-phenyl}-piperazine-1-carbaldehyde |
50994366 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Azd-4547 |
51039095 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
Torin 2 |
51358113 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
methyl 4-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzoate |
52941228 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzoic acid |
52942437 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(5-amino-3-(3-(dimethylamino)phenylamino)-1H-1,2,4-triazol-1-yl)(2,6-difluorophenyl)methanone |
52943663 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
ethyl 3-(5-amino-1-(2-fluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzoate |
52943672 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
ethyl 3-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzoate |
52944839 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-(5-amino-1-(2,6-difluorobenzoyl)-1H-1,2,4-triazol-3-ylamino)benzenesulfonamide |
52947304 |
ChemBL, TTD |