| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
3-(diethylamino)-N-[(16E)-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(24),2(27),3,5,8,10,12(26),16,21(25),22-decaen-10-yl]propanamide |
53363245 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-3-fluoro-11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(24),2(27),3,5,8(26),9,11,16,21(25),22-decaene |
53363246 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-23-fluoro-11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(24),2(27),3,5,8(26),9,11,16,21(25),22-decaene |
53363337 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-22-methoxy-11-(2-pyrrolidin-1-ylethoxy)-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8(26),9,11,16,21,23-decaene |
53363338 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-13,20-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8(26),9,11,16,21,23-decaene |
53364335 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-11-methoxy-14,19-dioxa-5,7,27-triazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(24),2(27),3,5,8(26),9,11,16,21(25),22-decaene |
53364337 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(E)-6,11-Dioxa-3-aza-2(4,2)-pyrimidina-1,4(1,3)-dibenzenacyclododecaphan-8-en-44-ol |
53364338 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2,6-dichlorophenyl)-N-(6-morpholin-4-ylpyrimidin-4-yl)-1H-imidazo[4,5-c]pyridin-4-amine |
53373594 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Itacitinib |
53380437 |
Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)-1-methylimidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide |
53475998 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)-3-methylimidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide |
53476000 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2,6-dichlorophenyl)-N-pyrimidin-4-yl-1H-imidazo[4,5-c]pyridin-4-amine |
53476104 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-Amino-N-Methyl-2-[4-(Morpholin-4-Yl)phenyl]thieno[3,2-C]pyridine-7-Carboxamide |
53497571 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-Amino-2-[4-(Tert-Butylsulfamoyl)phenyl]-N-Methylthieno[3,2-C]pyridine-7-Carboxamide |
53497572 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Jak-IN-1 |
54589404 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
2-((4-(4-Hydroxypiperidin-1-Yl)phenyl)amino)-5,11-Dimethyl-5h-Benzo[e]pyrimido [5,4-B][1,4]diazepin-6(11h)-One |
54592204 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
9-cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamine |
54760383 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
5-Chloro-4-(1H-indol-3-yl)-N-(2-methoxy-4-(4-(4-methylpiperazin-1-yl)piperidin-1-yl)phenyl)pyrimidin-2-amine |
56655374 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
Infigratinib Phosphate |
56669626 |
Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
(S)-(4-Fluorophenyl)(4-((5-methyl-1H-pyrazol-3-yl)amino)quinazolin-2-yl)methanol |
56833308 |
ChemBL |