| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
N-(2-(2,6-Dichlorophenyl)thiazolo[5,4-c]pyridin-4-yl)cyclopropanecarboxamide |
56953110 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-(2-(2,6-dichlorophenyl)thiazolo[4,5-d]pyrimidin-7-yl)cyclopropanecarboxamide |
56953203 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
{3,5-Dichloro-4-[4-(6-methyl-pyrimidin-4-ylamino)-thiazolo[5,4-c]pyridin-2-yl]-phenyl}-methanol |
56953205 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
1-(2-(2-Chloro-6-fluorophenyl)thiazolo[5,4-c]pyridin-4-yl)-3-cyclopropylurea |
56953296 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-(2-(2,6-Dichlorophenyl)thiazolo[5,4-c]pyridin-4-yl)-2-hydroxyacetamide |
56953392 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Cerdulatinib Hydrochloride |
56960607 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
1-(1-Benzylpiperidin-4-Yl)-1,6-Dihydroimidazo[4,5-D]pyrrolo[2,3-B]pyridine |
56973425 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-[4-[(4-Ethyl-1-piperazinyl)methyl]-3-(trifluoromethyl)anilino]-5,11-dimethyl-6-pyrimido[4,5-b][1,4]benzodiazepinone |
57340671 |
DSigDB |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-14-oxa-5,7,19,28-tetrazapentacyclo[17.5.2.12,6.18,12.022,26]octacosa-1(25),2(28),3,5,8,10,12(27),16,20,22(26),23-undecaene |
57342178 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(16E)-3-methyl-11-(2-pyrrolidin-1-ylethoxy)-14-oxa-5,7,19,28-tetrazapentacyclo[17.5.2.12,6.18,12.022,26]octacosa-1(25),2(28),3,5,8(27),9,11,16,20,22(26),23-undecaene |
57342180 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Peficitinib |
57928403 |
ChemBL, DGidb, GtoPDB, Pubchem, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(5-Hydroxyadamantan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
57928435 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(2r)-N-[4-[2-[(4-Morpholin-4-Ylphenyl)amino]pyrimidin-4-Yl]phenyl]pyrrolidine-2-Carboxamide |
57991377 |
TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-cyclohexyl-6H-isoxazolo[4,5-d]pyrrolo[2,3-b]pyridine |
58009815 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-Cyclohexyl-3-methyl-3,6-dihydropyrazolo[4,3-d]pyrrolo[2,3-b]pyridine |
58009825 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-Cyclohexyl-3,6-dihydropyrazolo[4,3-d]pyrrolo[2,3-b]pyridine |
58010054 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
5-amino-N-[2-(2,5-dichlorophenyl)pyrazol-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
58063089 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
5-amino-N-[3-(2,5-dimethylphenyl)-1-methylpyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
58063100 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
5-amino-N-[2-(5-chloro-2-methylphenyl)-5-methylpyrazol-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide |
58063103 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
5-Amino-pyrazolo[1,5-a]pyrimidine-3-carboxylic acid (2-methyl-4-o-tolyl-thiazol-5-yl)-amide |
58063108 |
ChemBL |