| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
JAK3 covalent inhibitor-1 |
137321159 |
DGidb, GtoPDB |
| TYK2 |
HGNC:12440 |
P29597 |
JAK3 inhibitor 34 |
137321160 |
DGidb, GtoPDB |
| TYK2 |
HGNC:12440 |
P29597 |
[(1S)-1-methyl-6-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydroinden-1-yl]cyanamide |
137349398 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Zasocitinib |
137441492 |
DGidb, GtoPDB |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)-[1,3]oxazolo[5,4-c]pyridin-4-yl]cyclopropanecarboxamide |
137631461 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[3-[(2-Cyanoacetyl)amino]phenyl]methylamino]pyrrolo[1,2-b]pyridazine-3-carboxamide |
137633211 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[[(3S)-3-methyl-1,1-dioxo-2,3-dihydro-1,2-benzothiazol-5-yl]amino]pyrazole-4-carboxamide |
137633780 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-ethyl-4-[3-(5-methyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl)-1H-indazol-6-yl]phenol |
137634328 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-(3,4-dicyanoanilino)pyrazole-4-carboxamide |
137634461 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-hydroxy-7-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]heptanamide |
137635398 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3,5-dichloro-4-[4-[[6-(methylamino)pyrimidin-4-yl]amino]-1H-imidazo[4,5-c]pyridin-2-yl]benzonitrile |
137635710 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[3-[[2-(3-Oxo-1,2-benzothiazol-2-yl)acetyl]amino]phenyl]methylamino]pyrrolo[1,2-b]pyridazine-3-carboxamide |
137637573 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-ethyl-4-[3-(5-methylsulfonyl-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-2-yl)-1H-indazol-6-yl]phenol |
137638897 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
[(3R)-3-(3-hydroxyphenyl)sulfonylpyrrolidin-1-yl]-[(3R,4R)-4-methyl-3-[methyl(7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl]methanone |
137642141 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-(3-chloro-4-cyanoanilino)-1-[(3R,4S)-4-cyanooxan-3-yl]pyrazole-4-carboxamide |
137642404 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)-3H-imidazo[4,5-c]pyridin-6-yl]cyclopropanecarboxamide |
137642443 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[(8-fluoro-4-methoxyquinolin-6-yl)amino]pyrazole-4-carboxamide |
137642740 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(1H-benzimidazol-2-yl)-1H-indazol-6-yl]-3-propan-2-ylphenol |
137643608 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-ethyl-4-[3-(1H-imidazol-2-yl)-1H-indazol-6-yl]phenol |
137645020 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)-[1,3]oxazolo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide |
137646825 |
ChemBL, TTD |