| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2,6-dichlorophenyl)isoquinolin-3-yl]cyclopropanecarboxamide |
137647912 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-[(4-chloro-8-fluoroquinolin-6-yl)amino]-1-[(3R,4S)-4-cyanooxan-3-yl]pyrazole-4-carboxamide |
137649981 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[4-(1-methylpyrazol-4-yl)anilino]pyrazole-4-carboxamide |
137651256 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-(4-cyclopropylanilino)pyrazole-4-carboxamide |
137651481 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-(2-ethyl-4-hydroxyphenyl)-N-methyl-1H-indazole-3-carboxamide |
137651710 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[(4-methylquinazolin-6-yl)amino]pyrazole-4-carboxamide |
137652173 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-hydroxy-7-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]octanamide |
137654793 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[[2-(dimethylamino)-6-fluoropyridin-4-yl]amino]pyrazole-4-carboxamide |
137654900 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)thieno[2,3-c]pyridin-7-yl]cyclopropanecarboxamide |
137655154 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[4-(triazol-1-yl)anilino]pyrazole-4-carboxamide |
137656215 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[2-[6-(2-ethyl-4-hydroxyphenyl)-1H-indazol-3-yl]-3,4,6,7-tetrahydroimidazo[4,5-c]pyridin-5-yl]ethanone |
137656346 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(1H-benzimidazol-2-yl)-1H-indazol-6-yl]-3-propylphenol |
137656679 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(1H-benzimidazol-2-yl)-1H-indazol-6-yl]-5-ethyl-2-fluorophenol |
137657080 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-(4-fluoroanilino)pyrazole-4-carboxamide |
137658028 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[2-(2,6-dichlorophenyl)furo[2,3-c]pyridin-7-yl]cyclopropanecarboxamide |
137658102 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-(4-cyano-3-cyclopropylanilino)-1-[(3R,4S)-4-cyanooxan-3-yl]pyrazole-4-carboxamide |
137659037 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[(3R,4S)-4-cyanooxan-3-yl]-3-[4-(difluoromethoxy)anilino]pyrazole-4-carboxamide |
137660124 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2,6-dichlorophenyl)isoquinolin-1-yl]cyclopropanecarboxamide |
137661036 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-(2,6-dichlorophenyl)-N-[6-[4-(oxetan-3-yl)piperazin-1-yl]pyrimidin-4-yl]-1H-imidazo[4,5-c]pyridin-4-amine |
137662248 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-Cyano-3-[5-(3-Cyclohexyl-3,5,8,10-Tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-Pentaen-4-Yl)furan-2-Yl]-~{n},~{n}-Dimethyl-Prop-2-Enamide |
138108525 |
ChemBL, TTD |