| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
Tyk2-IN-12 |
138739713 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-N-methylpyridine-3-carboxamide |
138756256 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
Tyk2-IN-7 |
138911330 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]cyclopropanecarboxamide |
139387327 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-[1-(2,2-difluorocyclopropanecarbonyl)-2,5-dihydropyrrol-3-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide |
139387328 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]-2,2-difluorocyclopropane-1-carboxamide |
139387329 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-[1-(cyclopropanecarbonyl)-3,6-dihydro-2H-pyridin-4-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide |
139387332 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[5-[1-(1-fluorocyclopropanecarbonyl)-2,5-dihydropyrrol-3-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide |
139387333 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohexyl]-2,2-difluorocyclopropane-1-carboxamide |
139387334 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohexyl]-1-fluorocyclopropane-1-carboxamide |
139387335 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1S)-N-[(1S)-4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]-2,2-difluorocyclopropane-1-carboxamide |
139387341 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1S)-N-[(1R)-4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]-2,2-difluorocyclopropane-1-carboxamide |
139387342 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1R)-N-[(1S)-4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]-2,2-difluorocyclopropane-1-carboxamide |
139387343 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1R)-N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohexyl]-2,2-difluorocyclopropane-1-carboxamide |
139387345 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1S)-N-[4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohexyl]-2,2-difluorocyclopropane-1-carboxamide |
139387346 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
(1R)-N-[(1R)-4-[2-(cyclopropanecarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-5-yl]cyclohex-3-en-1-yl]-2,2-difluorocyclopropane-1-carboxamide |
139387591 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
Jak2/flt3-IN-1 |
139600335 |
ChemBL, Pubchem |
| TYK2 |
HGNC:12440 |
P29597 |
8-(Cyclopropylamino)-6-(phenylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
140943115 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
8-(Cyclobutylamino)-6-[(3,5-dimethylphenyl)amino]imidazo[1,2-b]pyridazine-3-carboxamide |
140943118 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(3,5-Dimethylphenyl)amino]-8-(ethylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
140943126 |
ChemBL, TTD |