| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(3,5-Dimethylphenyl)amino]-8-(phenylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
140943142 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-([1,1'-Biphenyl]-3-ylamino)-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
140943145 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-(Cyclohexylamino)-8-(cyclopropylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
140943149 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
3-Methyl-4-phenyl-2,7-dihydropyrazolo[3,4-b]pyridin-6-one |
141335958 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
1-[3-[4-Amino-3-(1-methylpyrazol-4-yl)pyrazolo[3,4-d]pyrimidin-1-yl]pyrrolidin-1-yl]prop-2-en-1-one |
141531440 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[3-[[4-Amino-3-(1-methylpyrazol-4-yl)pyrazolo[3,4-d]pyrimidin-1-yl]methyl]piperidin-1-yl]prop-2-en-1-one |
141531442 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-[3-[4-Amino-3-(1-methylpyrazol-4-yl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one |
141531443 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[[5-chloro-4-(4-chloroanilino)pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728817 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[[7-[(2-fluorophenyl)methyl]pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728823 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-[4-[[7-[(2-fluorophenyl)methyl]pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyhexanamide |
141728826 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[[5-chloro-4-(cyclopropylamino)pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728840 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[[5-chloro-4-(3-chloroanilino)pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728841 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[[7-[(3-fluorophenyl)methyl]pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728858 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
7-[4-[(5-chloro-4-piperidin-1-ylpyrimidin-2-yl)amino]pyrazol-1-yl]-N-hydroxyheptanamide |
141728860 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[4-[[7-[(3-fluorophenyl)methyl]pyrrolo[2,3-d]pyrimidin-2-yl]amino]pyrazol-1-yl]-N-hydroxyhexanamide |
141728875 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(1-benzylpiperidin-4-yl)amino]-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
142753445 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(1-benzylpiperidin-4-yl)amino]-N-cyclopropyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
142753452 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[1-[(3-cyanophenyl)methyl]piperidin-4-yl]amino]-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
142753453 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[1-[(3-methoxyphenyl)methyl]piperidin-4-yl]amino]-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
142753457 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[1-[(2-methoxyphenyl)methyl]piperidin-4-yl]amino]-N-methyl-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
142753459 |
ChemBL |