| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-Carbamoylanilino)-6-[(5-fluoropyridin-2-yl)amino]pyridine-3-carboxamide |
154701267 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-6-[[1-[4-(2-hydroxypropan-2-yl)phenyl]-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155510753 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-6-[[1-(3-fluoropyridin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155510943 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[4-[(1R,4R)-5-(2-cyanoacetyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-2-yl]amino]-N-ethylbenzamide |
155510967 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[2-methoxy-3-(4-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridine-3-carboxamide |
155511037 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[4-[4-(2-cyanoacetyl)piperazin-1-yl]pyrimidin-2-yl]amino]-N-ethylbenzamide |
155511850 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-6-[[1-(5-fluoropyrimidin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155512660 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
8-(methylamino)-6-[(2-oxo-1-pyridin-2-ylpyridin-3-yl)amino]-N-propan-2-ylimidazo[1,2-b]pyridazine-3-carboxamide |
155513034 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[3-(2-hydroxyethylcarbamoyl)-2-methoxyanilino]-N-methylpyridine-3-carboxamide |
155513894 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[(1R,2S)-2-fluorocyclopropyl]-6-[[1-(5-fluoropyridin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155514076 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-Methylpropylamino)-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamide |
155514311 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[(1R)-1-cyclopropyl-1,3-dihydroxypropan-2-yl]amino]-6-(6-methoxypyridin-3-yl)pyrrolo[1,2-b]pyridazine-3-carboxamide |
155514805 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(ethylcarbamoyl)-2-methoxyanilino]-6-[(5-fluoro-4-methylpyridin-2-yl)amino]-N-methylpyridine-3-carboxamide |
155515726 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-8-(methylamino)-6-[[1-(6-methylpyridazin-3-yl)-2-oxopyridin-3-yl]amino]imidazo[1,2-b]pyridazine-3-carboxamide |
155516134 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoropyridin-2-yl)amino]-4-(2-methylsulfonylanilino)-N-(trideuteriomethyl)pyridine-3-carboxamide |
155517004 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
TYK2 inhibitor 47 |
155517088 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-methoxypyridin-2-yl)amino]-N-methyl-4-(2-methylsulfonylanilino)pyridine-3-carboxamide |
155517469 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
5-[[4-[(1R,5R)-8-(cyclopropanecarbonyl)-3,8-diazabicyclo[3.2.1]octan-3-yl]-5-fluoropyrimidin-2-yl]amino]-N-ethyl-3-methylpyridine-2-carboxamide |
155518120 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[(6-hydroxy-2-adamantyl)amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamide |
155518349 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[[4-[(1R,5R)-8-(cyclopropanecarbonyl)-3,8-diazabicyclo[3.2.1]octan-3-yl]-5-fluoropyrimidin-2-yl]amino]-N-ethylpyridine-3-carboxamide |
155520276 |
ChemBL, TTD |