| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoropyridin-2-yl)amino]-4-[2-methoxy-3-(methylcarbamoyl)anilino]-N-methylpyridine-3-carboxamide |
155538766 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(3-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155540191 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-carbamoylanilino)-6-[(5-fluoropyridin-2-yl)amino]-N,N-dimethylpyridine-3-carboxamide |
155540242 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155540484 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
methyl 3-[[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]sulfamoyl]propanoate |
155540621 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-8-(methylamino)-6-[(1-methyl-2-oxopyridin-3-yl)amino]imidazo[1,2-b]pyridazine-3-carboxamide |
155540954 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(1R,5R)-N-ethyl-3-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carboxamide |
155541097 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(3-chloro-4-hydroxyphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155541475 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-cyano-N-[4-[[[6-(4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]methyl]phenyl]acetamide |
155541478 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]cyclopentanesulfonamide |
155542401 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(1R,5R)-N-(cyanomethyl)-3-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carboxamide |
155542578 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]-1,1,1-trifluoromethanesulfonamide |
155542961 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
(1R,5R)-3-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-N-(2,2,2-trifluoroethyl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide |
155543349 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-[3-(cyclopropylmethylcarbamoyl)-2-methoxyanilino]-6-[(5-fluoro-4-methylpyridin-2-yl)amino]-N-methylpyridine-3-carboxamide |
155544232 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]pyridine-2-sulfonamide |
155545114 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]-2-piperidin-1-ylethanesulfonamide |
155545338 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-Fluoropyridin-2-yl)amino]-4-(2-methylsulfonylanilino)pyridine-3-carboxamide |
155546008 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(4-hydroxyphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155546232 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-methyl-6-(2-methylpropanoylamino)-4-(2-methylsulfonylanilino)pyridine-3-carboxamide |
155546437 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
cyclopropyl-[(1R,5R)-3-[5-fluoro-2-[[1-(2-hydroxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone |
155547916 |
ChemBL, TTD |