| GENE_SYMBOL |
HGNC_ID |
UNIPROT_ID |
DRUG_NAME |
PUBCHEM_CID |
Datasource |
| TYK2 |
HGNC:12440 |
P29597 |
4-[[4-[(1S,4S)-5-(cyclopropanecarbonyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-2-yl]amino]-N-ethylbenzamide |
155556520 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-6-[[1-(5-fluoropyridin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155558175 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-chloro-N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]benzenesulfonamide |
155558352 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
cyclopropyl-[(1R,5R)-3-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone |
155558729 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]pyridine-3-sulfonamide |
155559343 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
2-cyano-N-[3-[[[6-[[1-(2-methoxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]phenyl]acetamide |
155559609 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(4-hydroxy-3-methoxyphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155559746 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
5-(6-bromo-5-methoxy-1H-indol-3-yl)-2-(1H-pyrrol-2-yl)-1,3-oxazole |
155559898 |
ChemBL |
| TYK2 |
HGNC:12440 |
P29597 |
6-anilino-4-(2-carbamoylanilino)-N-methylpyridine-3-carboxamide |
155560352 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(4-hydroxy-2-methylphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155560413 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
cyclopropyl-[(1R,5R)-3-[5-fluoro-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone |
155561203 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
4-(2-carbamoylanilino)-6-[(3-fluoropyridin-2-yl)amino]-N-methylpyridine-3-carboxamide |
155561228 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-8-(methylamino)-6-[(2-oxo-1-pyridin-4-ylpyridin-3-yl)amino]imidazo[1,2-b]pyridazine-3-carboxamide |
155562327 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[(1R,2S)-2-fluorocyclopropyl]-6-[[1-(6-fluoropyridin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155563244 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[3-[[[6-[[1-(2-methoxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
155563799 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[3-[[[6-[[1-(2-hydroxyethyl)pyrazol-4-yl]amino]pyrimidin-4-yl]amino]methyl]phenyl]prop-2-enamide |
155564466 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-[6-(4-hydroxy-2,6-dimethylphenyl)-1H-indazol-4-yl]ethanesulfonamide |
155565077 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
N-cyclopropyl-6-[[1-(6-fluoropyridin-2-yl)-2-oxopyridin-3-yl]amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide |
155565275 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[2-methoxy-3-(2-morpholin-4-ylethylcarbamoyl)anilino]-N-methylpyridine-3-carboxamide |
155565520 |
ChemBL, TTD |
| TYK2 |
HGNC:12440 |
P29597 |
1-cyclobutyl-N-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-1H-indazol-4-yl]methanesulfonamide |
155565806 |
ChemBL, TTD |