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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACE H-Val-His-Leu-Ala-Pro-OH NA 4460000 NA NA NA NA BindingDB
ACE H-Leu-Ala-Leu-Pro-Pro-OH NA 794000000 NA NA NA NA BindingDB
ACE H-Val-Leu-Pro-Ile-Pro-OH NA 30900000 NA NA NA NA BindingDB
ACE H-Val-Arg-Gly-Pro-Phe-Pro-OH NA 588000000 NA NA NA NA BindingDB
ACE H-Asn-Ile-Phe-Tyr-Cys-Pro-OH NA 15100000 NA NA NA NA BindingDB
ACE H-Leu-His-Leu-Pro-Tyr-Pro-OH NA 2290000 NA NA NA NA BindingDB
ACE H-Leu-His-Leu-Pro-Gly-Pro-OH NA 1900000 NA NA NA NA BindingDB
ACE H-Leu-His-Leu-Tyr-Leu-Pro-OH NA 19000000 NA NA NA NA BindingDB
ACE H-Leu-His-Leu-Trp-Leu-Pro-OH NA 8910000 NA NA NA NA BindingDB
ACE L-Proline, L-valyl-L-tyrosyl- NA 288000000 NA NA NA NA BindingDB
ACE H-Ile-Arg-Pro-OH NA 741000 NA NA NA NA BindingDB
ACE L-Proline, L-valylglycyl- NA 26300000 NA NA NA NA BindingDB
ACE (5S)-5-[(N-benzoyl)amino]-4-oxo-6-phenyl-hexanoyl-L-tryptophan 195700 NA NA NA NA NA BindingDB|TTD
ACE 4-oxidanylidene-4-[[(2~{S})-1-oxidanyl-1-oxidanylidene-propan-2-yl]amino]butanoic acid NA 1348963|1348962.88 NA NA NA NA BindingDB|TTD
ACE (2S)-5-(diaminomethylideneamino)-2-(dithiolane-4-carbonylamino)pentanoic acid NA 113000 NA NA NA NA BindingDB|TTD
ACE [(3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl] dithiolane-4-carboxylate NA 347000 NA NA NA NA BindingDB|TTD
ACE Glycylglutamine NA 7079457.84 NA NA NA NA BindingDB|TTD
ACE Phe-Phe-Val-Ala-Pro NA 6020000 NA NA NA NA BindingDB
ACE Retrothiorphan NA 1000000000 NA NA NA NA TTD
ACE (3-Amino-2-oxo-azocan-1-yl)-acetic acid NA 440000 NA NA NA NA BindingDB|TTD