| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ZAP70 |
(5-{2-[1-(3-Carbamoyl-4-cyclohexylmethoxy-phenyl)-1-methyl-ethylcarbamoyl]-ethyl}-2-hydroxy-phenyl)-phosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
(S)-4-{(S)-2-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-propionylamino]-4-carboxy-butyrylamino}-4-((1S,2S)-1-carbamoyl-2-methyl-butylcarbamoyl)-butyric acid |
NA |
530000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
Ac-Tyr(PO3H2)-Asn-Glu-Leu-NH2 |
NA |
422000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
[4-[(2S)-2-acetamido-3-[[(1S)-4-amino-4-oxo-1-[3-[(4,6,6-trimethylcyclohexa-2,4-dien-1-yl)methyl]-1,2,4-oxadiazol-5-yl]butyl]amino]-3-oxopropyl]phenyl] dihydrogen phosphate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
Ac-Tyr(PO3H2)-Asp-Val-Leu-NH2 |
NA |
328000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
Src kinase inhibitor PP2 |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-{3-[(2,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
184000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ZAP70 |
4-[(2S)-2-{[(1S)-3-carbamoyl-1-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]propyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
4-[(2S)-2-acetamido-2-{[2-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)propan-2-yl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ZAP70 |
4-[(2S)-2-acetamido-2-{[(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ZAP70 |
4-[(2S)-2-acetamido-2-{[2-(3-{[4-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)ethyl]carbamoyl}ethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
4-[(2S)-2-{[(1S)-1-(3-benzyl-1,2,4-oxadiazol-5-yl)-3-carbamoylpropyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| ZAP70 |
1-[(3-Methyl-1-{2-[(1,2,3-Trimethyl-1h-Indol-5-Yl)amino]pyrimidin-4-Yl}-1h-Pyrazol-4-Yl)methyl]azetidin-3-Ol |
NA |
995800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |