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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
XDH 2-(4-Acetylanilino)-1-[4-(4-aminophenyl)piperazin-1-yl]ethanone NA 200000000 NA NA NA NA BindingDB
XDH 2-[4-(4-propan-2-yloxyphenyl)piperazine-1-carbonyl]-3H-benzimidazole-5-carboxamide NA 20000000000 NA NA NA NA BindingDB
XDH Monocerin NA 648000 NA NA NA NA TTD
XDH Nicotinic acid NA 518230 NA NA NA NA BindingDB|PubChem|TTD
XDH 2-Aminopurine NA 200000 NA NA NA NA TTD
XIAP (S)-N-((S)-2-((S)-2-(4-(4-fluoronaphthalen-1-yl)thiazol-2-yl)pyrrolidin-1-yl)-2-oxo-1-(tetrahydro-2H-pyran-4-yl)ethyl)-2-(methylamino)propanamide 140000 NA NA NA NA NA TTD
XIAP AoxSPY NA NA 120000 NA NA NA BindingDB
XIAP (2S,3R)-2-{[(2S)-1-({2-[(1S)-1-aminoethyl]-1,3-oxazol-4-yl}carbonyl)pyrrolidin-2-yl]formamido}-3-methylpentanoic acid NA NA 300000 NA NA NA BindingDB
XIAP (2S)-2-amino-N-[4-(2-chlorophenoxy)phenyl]propanamide NA NA 2e+05 NA NA NA ChEMBL
XIAP (S)-N-((S)-1-cyclohexyl-2-oxo-2-((S)-2-(7-phenylthiazolo[5,4-d]pyrimidin-2-yl)pyrrolidin-1-yl)ethyl)-2-(methylamino)propanamide 260000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-methylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-2-oxoethyl)-2-(methylamino)propanamide 940000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-isopropylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-2-oxoethyl)-2-(methylamino)propanamide 190000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-2-((S)-2-(4-benzylbenzo[d]thiazol-2-yl)pyrrolidin-1-yl)-1-cyclohexyl-2-oxoethyl)-2-(methylamino)propanamide 150000 NA NA NA NA NA TTD
XIAP (2S)-N-((1S)-2-((2S)-2-(4-(2-chlorophenyl)benzo[d]thiazol-2-yl)pyrrolidin-1-yl)-1-cyclohexyl-2-oxoethyl)-2-(methylamino)propanamide 160000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-1-cyclohexyl-2-oxo-2-((S)-2-(4-phenylthiazol-2-yl)pyrrolidin-1-yl)ethyl)-2-(methylamino)propanamide 190000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-3,3-dimethyl-1-oxo-1-((S)-2-(4-(quinolin-4-yl)thiazol-2-yl)pyrrolidin-1-yl)butan-2-yl)-2-(methylamino)propanamide 130000 NA NA NA NA NA TTD
XIAP (S)-N-((S)-2-((S)-2-(4-(benzo[d]isoxazol-3-yl)thiazol-2-yl)pyrrolidin-1-yl)-1-cyclohexyl-2-oxoethyl)-2-(methylamino)propanamide 120000 NA NA NA NA NA TTD
XIAP L-alanyl-L-valinamide NA 1200000 NA NA NA NA ChEMBL|TTD
XIAP (2S)-2-amino-N-(6-aminopyridin-2-yl)propanamide NA 110000 NA NA NA NA ChEMBL|TTD
XPNPEP1 2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolidin-1-yl]-4-phenyl-butyric acid NA 720000 NA NA NA NA BindingDB