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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC15A1
2-[[(2S)-2-amino-4-hydroxy-5-[(5-methyl-2,4-dioxopyrimidin-1-yl)methoxy]-5-oxopentanoyl]-methylamino]acetic acid
210000
NA
NA
NA
NA
NA
BindingDB
SLC15A1
2-[[(2R)-2-amino-3-(4-phenylmethoxyphenyl)propanoyl]amino]propanoic acid
1400000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
H-Pro-Asp-OH
NA|9800000
9160000|NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
Leucyl-glycyl-glycine
390000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
N-Methyl-L-alanyl-L-alanine
1800000
NA
NA
NA
NA
NA
TTD
SLC15A1
Ubenimex
400000
NA
NA
NA
NA
NA
BindingDB
SLC15A1
(2S)-2-[[(2S)-2-aminopropanoyl]amino]-3-(4-benzylphenyl)propanoic acid
120000
NA
NA
NA
NA
NA
TTD
SLC15A1
(2S)-1-[(2S)-2-amino-3-(1H-indol-2-yl)propanoyl]pyrrolidine-2-carboxylic acid
130000
NA
NA
NA
NA
NA
TTD
SLC15A1
(2S)-2-[[(2S)-2-amino-3-(1H-indol-2-yl)propanoyl]amino]propanoic acid
160000
NA
NA
NA
NA
NA
TTD
SLC15A1
Thr-Lys-Tyr
1100000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
Ile-Tyr
120000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
Pro-Ser
NA
NA
NA
1600000
NA
NA
BindingDB|TTD
SLC15A1
(2S)-2-[[(2S)-1-[(2S)-2-aminopropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoic acid
150000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
(2S)-6-amino-2-[[(2S)-3-phenyl-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoyl]amino]hexanoic Acid
2000000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
Leu-Leu
NA
170000
NA
NA
NA
NA
BindingDB|PubChem
SLC15A1
Oseltamivir Phosphate
NA
27400000
NA
NA
NA
NA
PubChem|TTD
SLC15A1
Leucylproline
180000|110000
NA
NA
NA
NA
NA
BindingDB|PubChem|TTD
SLC15A1
Leucyl-alanine
120000
NA
NA
NA
NA
NA
TTD
SLC15A1
Alanylproline
150000
NA
NA
NA
NA
NA
TTD
SLC15A1
NA
1400000
NA
NA
NA
NA
BindingDB
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