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HCDT 2.0
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negative DTIs
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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC15A2
Metampicillin
730000|724436|724435.96
NA
NA
NA
NA
NA
BindingDB|PubChem|TTD
SLC15A2
H-Pro-Asp-OH
2100000|2089296.13
NA
NA
NA
NA
NA
BindingDB|ChEMBL|TTD
SLC15A2
Prezatide
3100000|3090295.43|3090300
NA
NA
NA
NA
NA
BindingDB|ChEMBL|PubChem|TTD
SLC15A2
(2S)-6-amino-2-[[(2S)-3-phenyl-2-[[(2S)-pyrrolidine-2-carbonyl]amino]propanoyl]amino]hexanoic Acid
900000|891250.94
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A2
alanyl-D-alanine
270000|269153.48
NA
NA
NA
NA
NA
BindingDB|ChEMBL|TTD
SLC15A2
Prolyl-glycyl-glycine
11000000|10964781.96
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A2
Ala-Ala-Asp
160000|158489.32
NA
NA
NA
NA
NA
BindingDB|ChEMBL|TTD
SLC16A1
US10202350, Example 57
NA
133000
NA
NA
NA
NA
BindingDB
SLC16A1
US10202350, Example 56
NA
133000
NA
NA
NA
NA
BindingDB
SLC16A1
US10202350, Example 21
NA
300000
NA
NA
NA
NA
BindingDB
SLC16A1
US10202350, Example 22
NA
150000
NA
NA
NA
NA
BindingDB
SLC16A1
US10202350, Example 23
NA
300000
NA
NA
NA
NA
BindingDB
SLC16A1
US10202350, Example 49
NA
130000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-[(3-Methylquinolin-8-yl)sulfonylamino]phenyl]ethynyl]pyridine-2-carboxylic acid
NA
153000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-(Quinolin-8-ylsulfonylamino)phenyl]ethynyl]pyridine-2-carboxylic acid
NA
177000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-[(6-Methylquinolin-8-yl)sulfonylamino]phenyl]ethynyl]pyridine-2-carboxylic acid
NA
234000
NA
NA
NA
NA
BindingDB
SLC16A3
Mct4-IN-1
NA
638000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-[(4-Methylquinolin-8-yl)sulfonylamino]phenyl]ethynyl]pyridine-2-carboxylic acid
NA
209000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-[(2-Methylquinolin-8-yl)sulfonylamino]phenyl]ethynyl]pyridine-2-carboxylic acid
NA
245000
NA
NA
NA
NA
BindingDB
SLC16A3
5-[2-[2-[(5-Methylquinolin-8-yl)sulfonylamino]phenyl]ethynyl]pyridine-2-carboxylic acid
NA
283000
NA
NA
NA
NA
BindingDB
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