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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ABCB11 Dibenzothiophene NA 387900 NA NA NA NA TTD
ABCB11 3,6-diamino-N-[[(8Z)-15-amino-11-(2-amino-1,4,5,6-tetrahydropyrimidin-6-yl)-8-[(carbamoylamino)methylidene]-2-(hydroxymethyl)-3,6,9,12,16-pentaoxo-1,4,7,10,13-pentazacyclohexadec-5-yl]methyl]hexanamide NA 1000000 NA NA NA NA TTD
ABCB11 Diclofenac NA NA NA NA NA 300000 PubChem
ABCB11 Dolasetron methanesulfonate NA 133000 NA NA NA NA PubChem|TTD
ABCB11 (-)-(S)-9-Fluoro-2,3-dihydro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-7H-pyrido(1,2,3-de)-1,4-benzoxazine-6-carboxylic acid, hemihydrate NA 1000000|133000 NA NA NA NA PubChem
ABCB11 Gestodene NA 133000 NA NA NA NA PubChem|TTD
ABCB11 Orlistat NA 133000|NA NA NA NA NA|300000 PubChem|TTD
ABCB11 Quinine NA 135000|133000|NA NA NA NA NA|300000 PubChem
ABCB11 Dichlorphenamide NA 919100 NA NA NA NA PubChem|TTD
ABCB11 Choline NA NA NA NA NA 300000 PubChem
ABCB11 Prucalopride NA NA NA NA NA 300000 PubChem
ABCB11 Rasagiline Mesylate NA 133000 NA NA NA NA PubChem|TTD
ABCB11 Diflunisal NA NA NA NA NA 160000 PubChem
ABCB11 Capobenic acid NA 1000000 NA NA NA NA TTD
ABCB11 Diftalone NA 1000000 NA NA NA NA TTD
ABCB11 Fludarabine Phosphate NA 133000 NA NA NA NA PubChem|TTD
ABCB11 2-Aminohippuric acid NA 1000000 NA NA NA NA TTD
ABCB11 Dimethadione NA 1000000 NA NA NA NA TTD
ABCB11 Procromil NA 606000 NA NA NA NA TTD
ABCB11 Alclofenac NA NA NA NA NA 300000 PubChem