| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ALDH5A1 |
4-Hydroxybenzylamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ALDH5A1 |
4-Aminobenzoic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ALK |
Crizotinib |
NA |
380000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ALK |
5-chloro-4-N-(2-propan-2-ylsulfonylphenyl)-2-N-(5,6,7,8-tetrahydro-4H-[1,3]thiazolo[4,5-d]azepin-2-yl)pyrimidine-2,4-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ALK |
2-[[5-chloro-2-[[6-(2H-oxet-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-2-yl]amino]pyrimidin-4-yl]amino]-N-methylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ALK |
2-[[5-chloro-2-[[6-(oxetan-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-2-yl]amino]pyrimidin-4-yl]amino]-N-methylbenzamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ALK |
3-(5-Methyl-1H-pyrazol-3-yl)pyridine |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| ALK |
N-phenylquinolin-4-amine |
NA |
147000|112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| ALKBH2 |
(2R)-2-hydroxypentanedioic acid |
NA |
212000|424000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ALKBH2 |
(2S)-2-hydroxypentanedioic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
PubChem |
| ALKBH3 |
(2R)-2-hydroxypentanedioic acid |
NA |
8300000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ALKBH3 |
(2S)-2-hydroxypentanedioic acid |
NA |
24300000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| ALKBH3 |
N-(1-amino-3-methyl-1-oxobutan-2-yl)-4-(3-hydroxyphenyl)benzamide |
NA |
114600 |
NA |
NA |
NA |
NA |
BindingDB |
| ALKBH5 |
[2-(2-Chlorophenyl)pyrazolo[1,5-a]pyrimidin-6-yl]-(2-hydroxy-5-nitrophenyl)methanone |
NA |
101560 |
NA |
NA |
NA |
NA |
BindingDB |
| ALKBH5 |
ALKBH5 inhibitor DDO-2728 |
NA |
NA |
290300|373100 |
NA |
NA |
NA |
BindingDB |
| ALKBH5 |
3-[2-(4-Chlorophenyl)pyrazolo[1,5-a]pyrimidine-6-carbonyl]-4-hydroxybenzoic acid |
NA |
141470 |
NA |
NA |
NA |
NA |
BindingDB |
| ALKBH5 |
Citric Acid |
NA |
627900|488000 |
NA |
NA |
NA |
NA |
PubChem |
| ALKBH5 |
Ibuproxam, dimethyl deriv. |
NA |
135500|211100|269400 |
NA |
NA |
NA |
NA |
BindingDB |
| ALOX12 |
7-Ethyl-10-hydroxycamptothecin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| ALOX12 |
N-(5-butyramido-2-chlorophenyl)benzofuran-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |