| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| BCHE |
3-{3-[(Benzylmethylamino)methyl]phenyl}-6-methoxychromen-2-one |
NA |
136000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
3-{4-[(Benzylmethylamino)methyl]phenyl}-6-methoxychromen-2-one |
NA |
1300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
Trimethyl-[2-(pyridin-4-ylcarbamoyloxy)ethyl]azanium;iodide |
754200 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
N,N,N-trimethyl-2-(pyridin-4-ylcarbamoyloxy)ethanaminium iodide |
754200 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-[(2-Chloropyridin-4-yl)carbamoyloxy]ethyl-trimethylazanium;iodide |
161300 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
2-(2-chloropyridin-4-ylcarbamoyloxy)-N,N,N-trimethylethanaminium iodide |
161300 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-[(3-Bromopyridin-4-yl)carbamoyloxy]ethyl-trimethylazanium;iodide |
273800 |
NA |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
2-(3-bromopyridin-4-ylcarbamoyloxy)-N,N,N-trimethylethanaminium iodide |
273800 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(Dimethylamino)ethyl 2-chloropyridin-4-ylcarbamate dihydrochloride |
379700 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(Dimethylamino)ethyl 3-bromopyridin-4-ylcarbamate dihydrochloride |
273400 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| BCHE |
2-(Dimethylamino)ethyl 2,6-dichloropyridin-4-ylcarbamate hydrochloride |
174500 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
2-(Phenyl)-4-(3''-hydroxyphenyl)-2,3-dihydro-1,5-benzothiazepine |
NA |
142100|1421000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[[2-(Pyridin-1-ium-1-ylmethyl)phenyl]methyl]pyridin-1-ium;dibromide |
NA |
345000 |
NA |
NA |
NA |
NA |
TTD |
| BCHE |
Diacetyldistanol |
NA |
175800 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
((3S,3aS,4R,5R,7S,7aR)-3,3a,4-tris(benzyloxy)-7-methoxyhexahydro-2H-furo[2,3-c]pyran-5-yl)methanol |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
benzyl (2S)-2-[(3S,3aS,4R,5S,7S,7aR)-7-methoxy-3,3a,4-tris(phenylmethoxy)-2,3,4,5,7,7a-hexahydrofuro[2,3-c]pyran-5-yl]-2-hydroxyacetate |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[4-[4-(1-Hydroxycyclohexyl)triazol-1-yl]phenyl]ethanone |
NA |
450300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
(2E)-2-[[4-[[benzyl(methyl)amino]methyl]phenyl]methylidene]-5,6-dimethoxy-3H-inden-1-one |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
2-{4-[(Benzylmethylamino)methyl]benzylidene}-7-methoxy-3,4-dihydro-2H-naphthalen-1-one |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| BCHE |
1-[2-(2-Pyridin-1-ium-1-ylethoxy)ethyl]pyridin-1-ium;dibromide |
NA |
2360000 |
NA |
NA |
NA |
NA |
TTD |