Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CA2 | 4-amino-N-[4-(4-sulfamoylanilino)pyrimidin-2-yl]butanamide | 90907559.74 | NA | NA | NA | NA | NA | TTD |
| CA2 | 4-amino-N-(3-sulfamoylphenyl)butanamide | 5490000|5495408.74 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | 4-amino-N-(2-chloro-4-sulfamoylphenyl)butanamide | 32200000|32255219.38 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | N-{[(3aS,5aR,8aR,8bS)-2,2,7,7-tetramethyltetrahydro-3aH-bis[1,3]dioxolo[4,5-b:4',5'-d]pyran-3a-yl]methyl}sulfamide | 340000|650000 | NA | NA | NA | NA | NA | BindingDB |
| CA2 | 4-amino-N-(5-chloro-2,4-disulfamoylphenyl)butanamide | 111000000|111096403.5 | NA | NA | NA | NA|NA | NA|NA | BindingDB|TTD |
| CA2 | 4-amino-N-[4-[(4-sulfamoylphenyl)sulfamoyl]phenyl]butanamide | 71400000|71433182.62 | NA | NA | NA | NA|NA | NA|NA | BindingDB|TTD |
| CA2 | Syringic acid | 695000 | NA | NA | NA | NA | NA | BindingDB |
| CA2 | 7-Methoxycoumarin | 500000 | NA | NA | NA | NA | NA | TTD |
| CA2 | Coumarin-3-Carboxylic Acid | 500000 | NA | NA | NA | NA | NA | TTD |
| CA2 | Pyruvate | 2110000 | NA | NA | NA | NA | NA | BindingDB |
| CA2 | 4-amino-N-(2-fluoro-4-sulfamoylphenyl)butanamide | 99900000|100000000 | NA | NA | NA | NA|NA | NA|NA | BindingDB|TTD |
| CA2 | 4-amino-N-(2-bromo-4-sulfamoylphenyl)butanamide | 33300000|33334964.73 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | 4-[2-(4-Aminobutanoyl)hydrazinyl]benzenesulfonamide | 4720000|4716284.55 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | 4-amino-N-[3-oxo-3-[(5-sulfamoyl-1,3,4-thiadiazol-2-yl)amino]propyl]butanamide | 199986187 | NA | NA | NA | NA | NA | TTD |
| CA2 | 2-[(Dimethylamino)methyl]-4,5-dimethylphenol | NA | 880000 | NA | NA | NA | NA | BindingDB |
| CA2 | Selenic Acid | 112000000 | NA | NA | NA | NA | NA | PubChem|TTD |
| CA2 | 5-(4-Benzenesulfonyl-phenyl)-4-butyl-4H-[1,2,4]triazole-3-thiol | 604000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | Isothiocyanatosodium | 1600000 | NA | NA | NA | NA | NA | TTD |
| CA2 | trans-(1S(R),2S(R))-2-Hydroxycyclohexyl nitrate | 986000|NA | NA|560000 | NA | NA | NA | NA | BindingDB|TTD |
| CA2 | Sulfurous Acid | 8.9e+07|89000000 | NA | NA | NA | NA | NA | ChEMBL|TTD |