| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CA2 |
3-(4-(4-chlorophenylsulfonyl)phenyl)-4-propyl-1H-1,2,4-triazole-5(4H)-thione |
618000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA2 |
3-(4-(4-bromophenylsulfonyl)phenyl)-4-propyl-1H-1,2,4-triazole-5(4H)-thione |
382000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CA2 |
4-Methylpentanoate |
320000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
[Oxido(oxoboranyloxy)boranyl]oxy-oxoboranyloxyborinate |
950000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
Tetraborsaure |
950000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
Sodium Tetrafluoroborate |
100000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
|
48500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
|
570000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
|
920000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
|
950000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
|
112000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
7-(3-aminopyrrolidin-1-yl)-6-fluoro-3-[(3-phenylpropylamino)methyl]-1H-1,8-naphthyridin-4-one |
63000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
6-fluoro-3-(hydroxymethyl)-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
73000000|85000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
3-[(benzylamino)methyl]-6-fluoro-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
1600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
6-fluoro-7-pyrrolidin-1-yl-1H-1,8-naphthyridin-4-one |
89000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| CA2 |
6-(2-Sulfamoylbenzoyl)pyridine-2-carboxylic acid |
3571083.46 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
6-(2-Bromo-4-sulfamoylbenzoyl)pyridine-2-carboxylic acid |
32232945.95 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
6-(5-Chloro-2,4-disulfamoylbenzoyl)pyridine-2-carboxylic acid |
111173172.7 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
4,6-Diamino-5-chlorobenzene-1,3-disulfonamide |
35710834.58 |
NA |
NA |
NA |
NA |
NA |
TTD |
| CA2 |
6-(4-Sulfamoylbenzoyl)pyridine-2-carboxylic acid |
7575302.85 |
NA |
NA |
NA |
NA |
NA |
TTD |