GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ABCB11 |
(3E)-N-(4-chlorophenyl)-3-isopropylimino-5-(p-tolyl)phenazin-2-amine |
NA |
134900 |
NA |
NA |
NA |
NA |
TTD |
ABCB11 |
Voriconazole |
NA |
133000|NA |
NA |
NA |
NA |
NA|300000 |
PubChem|TTD |
ABCB11 |
Betamipron |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCB11 |
Synephrine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
Lorlatinib |
NA |
NA |
NA |
NA |
NA |
120000 |
PubChem |
ABCB11 |
Propylparaben |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
ABCB11 |
Alfuzosin Hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
Aceclofenac |
NA |
105000|NA |
NA |
NA |
NA |
NA|129999 |
PubChem|TTD |
ABCB11 |
Probicromil |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
ABCB11 |
Epanolol |
NA |
244400 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
N-[1,2-dimethoxy-10-methylsulfanyl-9-oxo-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]oxy-6,7-dihydro-5H-benzo[a]heptalen-7-yl]acetamide |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCB11 |
Levomepromazine |
NA |
127000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
H-Gly-Gly-Gly-Cys(1)-Tyr-Phe-Gln-Asn-Cys(1)-Pro-Lys-Gly-NH2.CH3CO2H |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
Doripenem |
NA |
133000|NA |
NA |
NA |
NA |
NA|300000 |
PubChem|TTD |
ABCB11 |
8-[4-methyl-3-[(5Z)-5-[(Z)-[5-[[2-methyl-5-[(4,6,8-trisulfo-2H-naphthalen-1-ylidene)carbamoyl]cyclohexa-2,4-dien-1-ylidene]carbamoyl]cyclohexa-2,4-dien-1-ylidene]carbamoyl]iminocyclohexa-1,3-diene-1-carbonyl]iminocyclohexa-1,4-diene-1-carbonyl]imino-7H-naphthalene-1,3,5-trisulfonic acid |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCB11 |
(1S,2R)-2-phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amine |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
ABCB11 |
Pyridostigmine Bromide |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
ABCB11 |
Histamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
Rizatriptan Benzoate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCB11 |
Oseltamivir Phosphate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |