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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ABCB11 (3E)-N-(4-chlorophenyl)-3-isopropylimino-5-(p-tolyl)phenazin-2-amine NA 134900 NA NA NA NA TTD
ABCB11 Voriconazole NA 133000|NA NA NA NA NA|300000 PubChem|TTD
ABCB11 Betamipron NA 133000 NA NA NA NA TTD
ABCB11 Synephrine NA 1000000 NA NA NA NA PubChem|TTD
ABCB11 Lorlatinib NA NA NA NA NA 120000 PubChem
ABCB11 Propylparaben NA NA NA NA NA 300000 PubChem
ABCB11 Alfuzosin Hydrochloride NA 133000 NA NA NA NA PubChem|TTD
ABCB11 Aceclofenac NA 105000|NA NA NA NA NA|129999 PubChem|TTD
ABCB11 Probicromil NA 1000000 NA NA NA NA TTD
ABCB11 Epanolol NA 244400 NA NA NA NA PubChem|TTD
ABCB11 N-[1,2-dimethoxy-10-methylsulfanyl-9-oxo-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]oxy-6,7-dihydro-5H-benzo[a]heptalen-7-yl]acetamide NA 133000 NA NA NA NA TTD
ABCB11 Levomepromazine NA 127000 NA NA NA NA PubChem|TTD
ABCB11 H-Gly-Gly-Gly-Cys(1)-Tyr-Phe-Gln-Asn-Cys(1)-Pro-Lys-Gly-NH2.CH3CO2H NA 133000 NA NA NA NA PubChem|TTD
ABCB11 Doripenem NA 133000|NA NA NA NA NA|300000 PubChem|TTD
ABCB11 8-[4-methyl-3-[(5Z)-5-[(Z)-[5-[[2-methyl-5-[(4,6,8-trisulfo-2H-naphthalen-1-ylidene)carbamoyl]cyclohexa-2,4-dien-1-ylidene]carbamoyl]cyclohexa-2,4-dien-1-ylidene]carbamoyl]iminocyclohexa-1,3-diene-1-carbonyl]iminocyclohexa-1,4-diene-1-carbonyl]imino-7H-naphthalene-1,3,5-trisulfonic acid NA 133000 NA NA NA NA TTD
ABCB11 (1S,2R)-2-phenylcyclopropan-1-amine;(1R,2S)-2-phenylcyclopropan-1-amine NA NA NA NA NA 300000 PubChem
ABCB11 Pyridostigmine Bromide NA 1000000 NA NA NA NA PubChem
ABCB11 Histamine NA 1000000 NA NA NA NA PubChem|TTD
ABCB11 Rizatriptan Benzoate NA 133000 NA NA NA NA PubChem|TTD
ABCB11 Oseltamivir Phosphate NA 133000 NA NA NA NA PubChem|TTD