| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| CHRNA4 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
8-Azabicyclo[3.2.1]octane, 2-[3-(4-chlorophenyl)-5-isoxazolyl]-8-methyl-3-(4-methylphenyl)-, (1R,2S,3S,5S)- |
NA |
942000 |
NA |
NA |
NA |
NA |
TTD |
| CHRNA4 |
4-Bromo-3-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-pyridine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CHRNA4 |
(1S,2R,4R,12S,15S,18R)-14,14,18-trimethyl-5,13-diazahexacyclo[13.3.1.02,13.04,12.04,18.06,11]nonadeca-6,8,10-trien-16-one |
NA |
145000 |
NA |
NA |
NA |
NA |
TTD |
| CHRNA4 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
2-Bromo-3-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-pyridine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CHRNA4 |
2-((R)-1-Methyl-pyrrolidin-2-yl)-furo[3,2-b]pyridine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| CHRNA4 |
1-(3-(Dimethylamino)butyl)-3-phenylurea |
316228|300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| CHRNA4 |
(5S)-spiro[1,3-oxazolidine-5,3'-1-azabicyclo[2.2.2]octane]-2-one |
NA |
2000000 |
NA |
NA |
NA |
NA |
TTD |
| CHRNA4 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| CHRNA4 |
Desformylflustrabromine |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| CHRNA4 |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| CHRNA4 |
Tropisetron |
NA |
170000 |
NA |
NA |
NA |
NA |
PubChem |
| CHRNA4 |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| CHRNA4 |
[(2S)-1-methylpyrrolidin-2-yl]methyl 3-aminobenzoate |
NA |
480000 |
NA |
NA |
NA |
NA |
BindingDB |
| CHRNA7 |
7-Methoxy-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,2-h]isoquinoline |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| CHRNA7 |
desformylflustrabromine-B |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |