| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| ABCB11 |
7-Chloro-2,3-dihydro-2-(4-methoxy-2-methylphenyl)pyridazino[4,5-b]quinoline-1,4,10(5H)-trione |
NA |
490000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
Semagacestat |
NA |
471900 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
(R)-2-(3-(Diisopropylamino)-1-phenylpropyl)-4-methylphenol 2,3-dihydroxysuccinate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Fesoterodine Fumarate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Cangrelor |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Rivaroxaban |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Fluorometholone |
NA |
100900 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
2-(furan-2-yl)-5-N-(2-morpholin-4-ylethyl)-[1,2,4]triazolo[1,5-a][1,3,5]triazine-5,7-diamine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
Pantolactone, (+/-)- |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
5-Chloro-2-methyl-2,3,3a,12b-tetrahydrodibenzo(2,3:6,7)oxepino(4,5-c)pyrrole |
NA |
NA |
NA |
NA |
NA |
269998 |
PubChem |
| ABCB11 |
(3R)-3-methyl-4-[4-(4-pyridin-4-ylpiperazin-1-yl)phenoxy]butanoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| ABCB11 |
(E)-But-2-enedioic acid;N-[2-hydroxy-5-[1-hydroxy-2-[1-(4-methoxyphenyl)propan-2-ylamino]ethyl]phenyl]formamide |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
Thiocolchicoside |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem |
| ABCB11 |
Tofacitinib |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCB11 |
2,2'-Azanediylbis(1-(6-fluorochroman-2-yl)ethanol) hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCC1 |
2-(3-Methyl-3-phenylthioureido)benzoic Acid |
NA |
198000 |
NA |
NA |
NA |
NA |
TTD |
| ABCC1 |
2-(4-Benzylpiperazine-1-carbonyl)-5-phenylmethoxychromen-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| ABCC2 |
Pazopanib |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCC2 |
Moxifloxacin Hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| ABCC2 |
Emetine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |