Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CTSD | US10246429, Example 344 | NA | 227000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 296 | NA | 289500 | NA | NA | NA | NA | BindingDB |
| CTSD | US10246429, Example 355 | NA | 141000 | NA | NA | NA | NA | BindingDB |
| CTSD | US9611261, Example 321 | NA | 212500 | NA | NA | NA | NA | BindingDB |
| CTSD | US9611261, Example 261 | NA | 444000 | NA | NA | NA | NA | BindingDB |
| CTSD | US9611261, Example 411 | NA | 359770 | NA | NA | NA | NA | BindingDB |
| CTSD | 2-amino-7-[4-(2-phenylethyl)phenyl]-3-[[(2S,5R)-5-phenyloxolan-2-yl]methyl]quinazolin-4-one | NA | 220000 | NA | NA | NA | NA | TTD |
| CTSD | 2-Amino-7-phenyl-3-[(4-phenyloxolan-2-yl)methyl]quinazolin-4-one | NA | 200000 | NA | NA | NA | NA | TTD |
| CTSD | N-[2-amino-7'-(3,6-dihydro-2H-pyran-5-yl)spiro[5H-1,3-oxazole-4,9'-xanthene]-2'-yl]-5-chloropyridine-2-carboxamide | NA | 470000 | NA | NA | NA | NA | BindingDB|TTD |
| CTSD | US10947223, Example 109 | NA | 1186500 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 104 | NA | 204000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 110 | NA | 524200 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 112 | NA | 970500 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 274 | NA | 122000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 113 | NA | 233000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 115 | NA | 119000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 183 | NA | 261000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 159 | NA | 143000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 139 | NA | 223000|428200|697800 | NA | NA | NA | NA | BindingDB |
| CTSD | US10947223, Example 105 | NA | 414900 | NA | NA | NA | NA | BindingDB |