Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CTSD | US11021493, Example 262 | NA | 108000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889581, Example 120 | NA | 190000 | NA | NA | NA | NA | BindingDB |
| CTSD | (3R)-3-[2-fluoro-5-[(Z)-2-fluoro-2-(5-prop-2-ynoxypyrazin-2-yl)ethenyl]phenyl]-3,6,6-trimethyl-1,1-dioxo-2H-1,4-thiazin-5-amine | NA | 230800 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 114 | NA | 115000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 138 | NA | 124600 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 244 | NA | 206000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 255 | NA | 122000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 239 | NA | 328800 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 124 | NA | 218000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 210 | NA | 467280 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 111 | NA | 107000|151000 | NA | NA | NA | NA | BindingDB |
| CTSD | US11021493, Example 181 | NA | 178000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 102 | NA | 211000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 107 | NA | 281800 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 103 | NA | 186000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 108 | NA | 385600 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 111 | NA | 300500 | NA | NA | NA | NA | BindingDB |
| CTSD | US11548903, Example 141 | NA | 237000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 104 | NA | 133000 | NA | NA | NA | NA | BindingDB |
| CTSD | US10889579, Example 113 | NA | 178000 | NA | NA | NA | NA | BindingDB |