GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
ABCC2 |
Olanzapine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Raltitrexed |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Allopurinol |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Leucovorin Calcium |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Sildenafil Citrate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Aprepitant |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Tegaserod Maleate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
1-(3-Chlorophenyl)piperazine |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Entecavir Hydrate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem |
ABCC2 |
4-(3-(3-(Ethoxycarbonyl)-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)thioureido)benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
ABCC2 |
CID 137648451 |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCC2 |
(1R,2R,3R,6R,7S,9R,10R,12R,13S,15R,17S)-9-[(2S,3R,4S,6R)-4-(dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-3-ethyl-2,10-dihydroxy-7-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-15-(2-methoxyethoxymethyl)-2,6,10,12,17-pentamethyl-4,16-dioxa-14-azabicyclo[11.3.1]heptadecan-5-one |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCC2 |
Ethambutol Hydrochloride |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
(2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-[(1S,2S,3R,4S,6R)-4,6-diamino-2-[(2S,3R,4S,5R)-4-[(2R,3R,4R,5S)-3-amino-6-(aminomethyl)-4,5-dihydroxyoxan-2-yl]oxy-3-hydroxy-5-(hydroxymethyl)oxolan-2-yl]oxy-3-hydroxycyclohexyl]oxyoxane-3,4-diol |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
ABCC2 |
Escitalopram Oxalate |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Rabeprazole Sodium |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Docetaxel |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Ezetimibe |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Lumiracoxib |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
ABCC2 |
Metylperon |
NA |
133000 |
NA |
NA |
NA |
NA |
PubChem|TTD |