Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| CYP1A2 | methyl N-[4-[(4-fluorophenyl)methyl-prop-2-ynyl-amino]-2,6-dimethyl-phenyl]carbamate | NA | 142000 | NA | NA | NA | NA | BindingDB |
| CYP1A2 | Naphthalene | NA | 700000 | NA | NA | NA | NA | BindingDB|PubChem |
| CYP1A2 | 1-Naphthalenyl[4-(pentyloxy)-1-naphthalenyl]methanone | NA | 200000 | NA | NA | NA | NA | PubChem |
| CYP1A2 | (E)-3,5,30,50-Tetramethoxystilbene | NA | 198000 | NA | NA | NA | NA | BindingDB |
| CYP1B1 | Alpha-Naphthoflavone | NA | 110600 | NA | NA | NA | NA | BindingDB |
| CYP1B1 | 4-[(e)-Phenyldiazenyl]morpholine | NA | 163000 | NA | NA | NA | NA | BindingDB|TTD |
| CYP1B1 | Fluoxetine | NA | 475000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CYP1B1 | Furafylline | 200000 | NA | NA | NA | NA | NA | TTD |
| CYP1B1 | Bergamottin | 587000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CYP1B1 | Testosterone | 411800 | NA | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| CYP1B1 | 4-Methoxyestradiol | 149000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| CYP1B1 | 4-[(E)-morpholin-4-yldiazenyl]benzoic acid | NA | 400000 | NA | NA | NA | NA | BindingDB|TTD |
| CYP1B1 | 4-Aminobenzoic Acid | NA | 120000 | NA | NA | NA | NA | PubChem|TTD |
| CYP24A1 | 2-Bromo-Benzylidene Tetralone | NA | 122000 | NA | NA | NA | NA | BindingDB|TTD |
| CYP24A1 | 2-(biphenyl-2-ylmethyl)-6-methoxy-3,4-dihydronaphthalen-1(2H)-one | NA | 127600 | NA | NA | NA | NA | BindingDB|TTD |
| CYP24A1 | 2-(2-(E)-Styrylbenzyl)-6-methoxy-tetralone | NA | 342800 | NA | NA | NA | NA | BindingDB|TTD |
| CYP24A1 | (E)-2-(biphenyl-2-ylmethylene)-6-methoxy-3,4-dihydronaphthalen-1(2H)-one | NA | 111100 | NA | NA | NA | NA | BindingDB|TTD |
| CYP24A1 | (2E)-6-Methoxy-2-[(2-methylphenyl)methylidene]-1,2,3,4-tetrahydronaphthalen-1-one | NA | 480100 | NA | NA | NA | NA | BindingDB|TTD |
| CYP2A13 | ethyl 3-(1H-imidazol-1-yl)propanoate | NA | 238000 | NA | NA | NA | NA | BindingDB |
| CYP2A13 | 2-Nonyl-1H-imidazole | NA | 277000 | NA | NA | NA | NA | BindingDB |