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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
CYP2B6 3-(4-Pyridin-3-ylpyridin-3-yl)prop-2-yn-1-amine;trihydrochloride NA 364000 NA NA NA NA TTD
CYP2B6 1-[(2R)-1-hydroxy-3-phenylpropan-2-yl]-2-methylpyridin-1-ium-3,4-diol;chloride NA 200000 NA NA NA NA TTD
CYP2B6 6-(Benzotriazol-1-ylamino)hexanoic acid NA 258000 NA NA NA NA TTD
CYP2B6 1-(5-(Pyridin-3-yl)thiophen-2-yl)ethan-1-one NA 217000 NA NA NA NA TTD
CYP2B6 3-(2-Methyl-1H-imidazol-1-yl)pyridine 300000 NA NA NA NA NA TTD
CYP2B6 5-Hydroxy saxagliptin NA 200000 NA NA NA NA TTD
CYP2B6 1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)-4-(4-(trifluoromethyl)phenyl)pyridin-2(1H)-one NA 10000000 NA NA NA NA TTD
CYP2B6 4-(2,4-dichlorophenyl)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one NA 10000000 NA NA NA NA TTD
CYP2B6 Carbamazepine NA NA NA 145000 NA NA PubChem|TTD
CYP2B6 3-(3-Methyl-1H-imidazol-4-yl)-pyridine NA 146000 NA NA NA NA TTD
CYP2B6 3-(4-Methyl-imidazol-1-yl)-pyridine NA 300000 NA NA NA NA TTD
CYP2B6 (5-Pyridin-3-ylthiophen-2-yl)methanamine;(5-pyridin-3-ylthiophen-2-yl)methanimine NA 256000 NA NA NA NA TTD
CYP2B6 1-[5-(4-Cyanophenyl)-2-bicyclo[3.1.0]hexanyl]-3-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[3-(4-methylpiperazin-1-yl)propyl]urea NA 10000000 NA NA NA NA TTD
CYP2B6 (NE)-N-[(5-pyridin-3-ylfuran-2-yl)methylidene]hydroxylamine;(NZ)-N-[(5-pyridin-3-ylfuran-2-yl)methylidene]hydroxylamine NA 206000 NA NA NA NA TTD
CYP2B6 Auglurant NA 200000 NA NA NA NA TTD
CYP2B6 3,3'-Bipyridine NA 145000 NA NA NA NA TTD
CYP2B6 Thieno[3,2-d]pyrimidin-4(3H)-one, 6-(4-chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]- NA 10000000 NA NA NA NA TTD
CYP2C18 4-methyl-N-(1-phenyl-1H-pyrazol-5-yl)benzenesulfonamide NA 170000 NA NA NA NA BindingDB
CYP2C18 4-Allyl-N-benzyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfonamide NA 125000 NA NA NA NA BindingDB
CYP2C18 4-Allyl-N-(2-phenyl-2H-pyrazol-3-yl)-benzenesulfonamide NA 150000 NA NA NA NA BindingDB